SCHEMBL7833601

SCHEMBL7833601

CCc1ccc2cc(NC=O)ccc2n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.39
RAB9A P51151 4/20 0.39
CCNE2 O96020 1/20 0.39
CDK4 P11802 1/20 0.39
CCND1 P24385 1/20 0.39
CCNE1 P24864 1/20 0.39
CDK2 P24941 1/20 0.39
KDM4E B2RXH2 2/20 0.35
LIPG Q9Y5X9 1/20 0.34
HDAC1 Q13547 3/20 0.33
HDAC2 Q92769 3/20 0.33
ALDH1A1 P00352 3/20 0.33
TERT O14746 2/20 0.33
GRM1 Q13255 1/20 0.33
GAA P10253 1/20 0.33
HTR2C P28335 1/20 0.33
MCHR1 Q99705 1/20 0.33
PDE10A Q9Y233 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10133371 0.79 NPC1 (0.52) NPC1RAB9ACCNE2CDK4CCND1
SCHEMBL9458481 0.78 CCNE2 (0.44) NPC1CCNE2CDK4CCND1CCNE1
SCHEMBL4586790 0.76 ALDH1A3 (0.39) HDAC1HDAC2ALDH1A1GAAPDE10A
SCHEMBL5959990 0.76 NMT1 (0.40) NPC1RAB9ACCNE2CDK4CCND1
SCHEMBL5873649 0.76 PLAU (0.52) MCHR1
SCHEMBL27689981 0.73 ALDH1A1 (0.50) NPC1RAB9ACCNE2CDK4CCND1
SCHEMBL28161952 0.71 LMNA (0.40) ALDH1A1MEN1KMT2A
SCHEMBL6230105 0.71 CYP1A2 (0.59) NPC1RAB9AKDM4EALDH1A1MEN1
SCHEMBL12824284 0.71 CYP1A2 (0.50) NPC1RAB9AKDM4EALDH1A1TERT
SCHEMBL9413345 0.70 LMNA (0.47) NPC1RAB9AALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5444071-A Hypotensive agent IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1995-08-22 US claimed
EP-0412848-B1 Quinoline derivatives, process for their preparation and their use as medicaments ICI PLC (GB) 1995-01-18 EP claimed
EP-0412848-A2 Quinoline derivatives, process for their preparation and their use as medicaments ZENECA LIMITED (GB) 1991-02-13 EP claimed
EP-0470795-B2 Process for the manufacture of nitriles AVECIA LTD (GB) 2001-02-21 EP disclosed
US-5444071-A Hypotensive agent IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1995-08-22 US disclosed
EP-0470794-B1 Process for the preparation of nitriles ZENECA LTD (GB) 1995-01-25 EP disclosed
EP-0470795-B1 Process for the manufacture of nitriles ZENECA LTD (GB) 1995-01-25 EP disclosed
EP-0412848-B1 Quinoline derivatives, process for their preparation and their use as medicaments ICI PLC (GB) 1995-01-18 EP disclosed
EP-0495948-A1 PROCESS FOR THE MANUFACTURE OF QUINOLINE DERIVATIVES ZENECA LIMITED (GB) 1992-07-29 EP disclosed
WO-1992002508-A1 PROCESS FOR THE MANUFACTURE OF QUINOLINE DERIVATIVES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-02-20 WO disclosed
EP-0470795-A1 Process for the manufacture of nitriles ZENECA LIMITED (GB) 1992-02-12 EP disclosed
EP-0470794-A1 Process for the preparation of nitriles ZENECA LIMITED (GB) 1992-02-12 EP disclosed
EP-0412848-A2 Quinoline derivatives, process for their preparation and their use as medicaments ZENECA LIMITED (GB) 1991-02-13 EP disclosed