SCHEMBL7833700

SCHEMBL7833700

O=C(O)COc1ccc(SCc2nc3ccc(-n4ccnc4)cc3[nH]2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CBFB Q13951 1/20 0.43
CYP3A4 P08684 3/20 0.41
CYP2D6 P10635 3/20 0.41
PORCN Q9H237 1/20 0.41
FGFR1 P11362 2/20 0.41
FLT1 P17948 1/20 0.41
TBXAS1 P24557 3/20 0.41
LMNA P02545 4/20 0.41
MAPK1 P28482 1/20 0.41
F9 P00740 1/20 0.40
GRK6 P43250 1/20 0.39
MAPT P10636 4/20 0.39
ALDH1A1 P00352 2/20 0.39
HTT P42858 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
HPGD P15428 1/20 0.39
FGFR2 P21802 1/20 0.39
FGFR3 P22607 1/20 0.39
RAB9A P51151 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7834577 0.85 CYP11B1 (0.51) CBFBCYP3A4CYP2D6FGFR1FLT1
SCHEMBL7832392 0.83 CBFB (0.47) CBFBCYP3A4CYP2D6FGFR1FLT1
SCHEMBL7821991 0.83 NPC1 (0.55) CBFBCYP3A4CYP2D6FGFR1FLT1
Hydrochloric Acid SCHEMBL8155594 0.82 NPC1 (0.54) CBFBCYP3A4CYP2D6FGFR1FLT1
SCHEMBL7822236 0.81 TNIK (0.45) CBFBFGFR1FLT1F9ALDH1A1
Hydrochloric Acid SCHEMBL8143148 0.81 TNIK (0.44) CBFBFGFR1FLT1F9ALDH1A1
SCHEMBL7833681 0.78 ADH5 (0.48) CBFBCYP3A4CYP2D6TBXAS1LMNA
SCHEMBL7834574 0.77 CYP11B1 (0.51) CBFBCYP3A4CYP2D6LMNAMAPK1
SCHEMBL7832389 0.76 ENPP2 (0.47) CBFBCYP3A4CYP2D6FGFR1FLT1
SCHEMBL7821732 0.75 RAB9A (0.58) CBFBCYP3A4CYP2D6FGFR1FLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0894795-B1 Benzimidazole, benzoxazole and benzothiazole derivatives, their preparation and pharmaceutical compositions containing them ADIR (FR) 2001-06-06 EP disclosed
US-6040327-A INHIBITORS OF INTERLEUKINS; TREATING RHEUMATOID ARTHRITIS OR ARTHROSIS ADIR ET COMPAGNIE (FR) 2000-03-21 US disclosed
EP-0894795-A1 Benzimidazole, benzoxazole and benzothiazole derivatives, their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1999-02-03 EP disclosed