SCHEMBL7833959

SCHEMBL7833959

OCc1nc2cccnc2n1Cc1ccc(-c2ccccc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.60
ENPP2 Q13822 11/20 0.54
TP53 P04637 2/20 0.53
TBXA2R P21731 1/20 0.52
AGTR1 P30556 2/20 0.52
AGTR2 P50052 2/20 0.52
MEN1 O00255 1/20 0.51
MAPT P10636 1/20 0.51
KMT2A Q03164 1/20 0.51
BRD4 O60885 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17966877 0.85 TP53 (0.62) LMNAENPP2TP53TBXA2RMAPT
SCHEMBL7095165 0.84 LMNA (0.54) LMNAENPP2TP53TBXA2RAGTR1
SCHEMBL15244777 0.78 LMNA (0.66) LMNAENPP2TP53TBXA2RMEN1
SCHEMBL7823224 0.76 LMNA (0.46) LMNAENPP2TP53TBXA2RMEN1
SCHEMBL9853648 0.76 PPARG (0.74) AGTR1AGTR2
SCHEMBL15071581 0.75 BRD4 (0.51) LMNAENPP2TP53TBXA2RAGTR1
SCHEMBL9760633 0.75 LMNA (0.61) LMNAENPP2TP53MEN1KMT2A
SCHEMBL7851373 0.74 AGTR1 (0.75) AGTR1AGTR2
SCHEMBL8566073 0.73 PPARG (0.61) LMNAENPP2TP53TBXA2RAGTR1
SCHEMBL9761791 0.73 LMNA (0.59) LMNAENPP2TP53TBXA2RMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0676398-B1 Heterocyclic compounds having anti-diabetic activity, their preparation and their use SANKYO CO (JP) 2001-10-24 EP disclosed
US-6117893-A Heterocyclic compounds having anti-diabetic activity and their use SANKYO COMPANY, LIMITED (JP) 2000-09-12 US disclosed
EP-1022274-A1 Oxazolidinedione and Thiazolidinedione derivatves, their preparation and their use Sankyo Company Limited (JP) 2000-07-26 EP disclosed
US-5977365-A HYPOGLYCEMIC AGENTS SANKYO COMPANY, LIMITED (JP) 1999-11-02 US disclosed
US-5962470-A Heterocyclic compounds having anti-diabetic activity and their use SANKYO COMPANY, LIMITED (JP) 1999-10-05 US disclosed
US-5834501-A TREATING DIABETES OR HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 1998-11-10 US disclosed
US-5739345-A HYPOGLYCEMIC AND ANTIDIABETIC AGENTS SANKYO COMPANY, LIMITED (JP) 1998-04-14 US disclosed
US-5624935-A ANTIDIABETIC AGENTS, HYPOGLYCEMIC AGENTS OR ANTILIPEMIC AGENTS SANKYO COMPANY, LIMITED 1997-04-29 US disclosed
EP-0676398-A2 Heterocyclic compounds having anti-diabetic activity, their preparation and their use SANKYO COMPANY LIMITED (JP) 1995-10-11 EP disclosed