SCHEMBL7834666

SCHEMBL7834666

COC(=O)CC1CCN(C(=O)C(C2CC2)C(C)(C)NC(=O)c2ccc(C#N)cc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.41
PRSS1 P07477 1/20 0.38
CTSG P08311 1/20 0.38
CTRB1 P17538 1/20 0.38
CMA1 P23946 1/20 0.38
CHRM4 P08173 1/20 0.38
GPR119 Q8TDV5 1/20 0.37
ITGB3 P05106 9/20 0.37
ITGA2B P08514 9/20 0.37
PDK2 Q15119 2/20 0.36
CCR3 P51677 1/20 0.36
PRKAB2 O43741 1/20 0.36
CYP3A4 P08684 1/20 0.36
PRKAG1 P54619 1/20 0.36
PRKAA2 P54646 1/20 0.36
PRKAA1 Q13131 1/20 0.36
PRKAG3 Q9UGI9 1/20 0.36
PRKAG2 Q9UGJ0 1/20 0.36
PRKAB1 Q9Y478 1/20 0.36
YAP1 P46937 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7825201 0.89 SIGMAR1 (0.43) SIGMAR1PRSS1CTSGCTRB1CMA1
SCHEMBL7834781 0.83 SIGMAR1 (0.37) SIGMAR1PRSS1CTSGCTRB1CMA1
SCHEMBL7837372 0.80 ITGB3 (0.45) SIGMAR1PRSS1CTSGCTRB1CMA1
SCHEMBL7835452 0.78 PRSS1 (0.44) SIGMAR1PRSS1CTSGCTRB1CMA1
SCHEMBL7836103 0.78 CTSG (0.43) PRSS1CTSGCTRB1CMA1CHRM4
SCHEMBL7825622 0.77 NPC1 (0.46) PRSS1CTSGCTRB1CMA1
SCHEMBL7836339 0.76 YAP1 (0.44) PRSS1CTSGCTRB1CMA1CHRM4
SCHEMBL7833800 0.76 YAP1 (0.44) PRSS1CTSGCTRB1CMA1CHRM4
SCHEMBL7833511 0.76 ITGB3 (0.65) ITGB3ITGA2B
SCHEMBL7833534 0.76 YAP1 (0.43) PRSS1CTSGCTRB1CMA1CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0800516-B1 FIBRINOGEN RECEPTOR ANTAGONISTS HAVING SUBSTITUTED (b)-AMINO ACID RESIDUES AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME NIPPON STEEL CORP (JP) 2001-09-19 EP disclosed
US-5866592-A Fibrinogen receptor antagonist and pharmaceutical compositions comprising the same NIPPON STEEL CORPORATION (JP) 1999-02-02 US disclosed