SCHEMBL7835970

SCHEMBL7835970

CC(C)(NC(=O)c1ccc(C#N)cc1)C(CC1CCCCC1)C(=O)N1CCC(CC(=O)OCc2ccccc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
YAP1 P46937 3/20 0.41
CHRM4 P08173 2/20 0.41
HTRA1 Q92743 1/20 0.40
CTSS P25774 7/20 0.40
CTSL P07711 4/20 0.40
CTSB P07858 4/20 0.40
CTSK P43235 2/20 0.40
CCR3 P51677 1/20 0.39
P2RX7 Q99572 1/20 0.37
PRSS1 P07477 1/20 0.37
CTSG P08311 1/20 0.37
CTRB1 P17538 1/20 0.37
CMA1 P23946 1/20 0.37
CCR1 P32246 1/20 0.36
PREP P48147 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7833800 0.91 YAP1 (0.44) YAP1CHRM4CCR3P2RX7PRSS1
SCHEMBL7838327 0.88 ITGB3 (0.48) PRSS1
SCHEMBL7836339 0.86 YAP1 (0.44) YAP1CHRM4CCR3P2RX7PRSS1
SCHEMBL7833534 0.86 YAP1 (0.43) YAP1CHRM4CTSLCTSBCTSK
SCHEMBL7835873 0.83 YAP1 (0.41) YAP1CHRM4CCR3P2RX7PRSS1
SCHEMBL7833217 0.83 GRIN2B (0.42) YAP1CHRM4CCR3P2RX7PRSS1
SCHEMBL7357897 0.82 YAP1 (0.46) YAP1CHRM4CCR3P2RX7PRSS1
SCHEMBL8791368 0.82 CHRM4 (0.44) YAP1CHRM4CCR3PRSS1CTSG
SCHEMBL7839324 0.82 ITGB3 (0.44) YAP1CHRM4CCR3P2RX7PRSS1
SCHEMBL7824541 0.81 CCR1 (0.51) YAP1CHRM4CCR3PRSS1CTSG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0800516-B1 FIBRINOGEN RECEPTOR ANTAGONISTS HAVING SUBSTITUTED (b)-AMINO ACID RESIDUES AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME NIPPON STEEL CORP (JP) 2001-09-19 EP disclosed
US-5866592-A Fibrinogen receptor antagonist and pharmaceutical compositions comprising the same NIPPON STEEL CORPORATION (JP) 1999-02-02 US disclosed