SCHEMBL7836686

SCHEMBL7836686

CCOC(=O)c1[nH]c2cc(Br)ccc2c1CC#N

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.46
MAPT P10636 4/20 0.46
ALOX15 P16050 4/20 0.46
GPR17 Q13304 1/20 0.45
HTR1A P08908 1/20 0.45
DRD2 P14416 1/20 0.45
DRD4 P21917 1/20 0.45
HTR1D P28221 1/20 0.45
HTR1B P28222 1/20 0.45
HTR1F P30939 1/20 0.45
HTR7 P34969 1/20 0.45
DRD3 P35462 1/20 0.45
GABRA1 P14867 1/20 0.43
GABRB1 P18505 1/20 0.43
GABRA3 P34903 1/20 0.43
GABRB2 P47870 1/20 0.43
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 3/20 0.43
NPSR1 Q6W5P4 2/20 0.43
NPC1 O15118 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7826411 0.86 HTR6 (0.46) HTR6MAPTALOX15GPR17HTR1A
SCHEMBL12326581 0.83 HTR6 (0.67) HTR6MAPTHTR1ADRD2DRD4
SCHEMBL2204200 0.82 HTR6 (0.53) HTR6MAPTALOX15GPR17HTR1A
SCHEMBL2202482 0.81 GPR17 (0.57) HTR6MAPTALOX15GPR17HTR1A
SCHEMBL24074581 0.81 ALDH1A1 (0.58) MAPTALOX15GPR17GABRA1GABRB1
SCHEMBL8795754 0.80 ALOX15 (0.61) MAPTALOX15
SCHEMBL20535547 0.79 ALOX15 (0.50) MAPTALOX15GPR17GABRA1GABRB1
SCHEMBL28477589 0.79 KDM4E (0.64) HTR6MAPTALOX15GABRA1GABRB1
SCHEMBL7838931 0.79 ALOX15 (0.46) HTR6MAPTALOX15HTR1ADRD2
SCHEMBL7834192 0.79 ALDH1A1 (0.60) MAPTALOX15ALDH1A1KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1147110-A1 PYRAZINO(AZA)INDOLE DERIVATIVES VERNALIS RESEARCH LIMITED (GB) 2001-10-24 EP disclosed
WO-2000044753-A1 PIRAZINO(AZA)INDOLE DERIVATIVES VERNALIS RESEARCH LIMITED (GB) 2000-08-03 WO disclosed