SCHEMBL7840740

SCHEMBL7840740

COC(=O)CNS(=O)(=O)Cl

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 7/20 0.52
CA14 Q9ULX7 5/20 0.52
CA2 P00918 4/20 0.52
TET2 Q6N021 1/20 0.46
GAA P10253 3/20 0.46
KDM4E B2RXH2 2/20 0.46
NPC1 O15118 1/20 0.46
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
RECQL P46063 1/20 0.45
TSHR P16473 5/20 0.42
EPHX2 P34913 1/20 0.40
HSD17B10 Q99714 2/20 0.39
MGAM O43451 1/20 0.39
SI P14410 1/20 0.39
MGAM2 Q2M2H8 1/20 0.39
CA9 Q16790 4/20 0.38
CA1 P00915 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3365530 0.80 GAA (0.50) GAANPC1ALDH1A1HPGDRAB9A
SCHEMBL14962838 0.80 CA12 (0.51) CA12CA14CA2GAAKDM4E
SCHEMBL8930152 0.78 CA12 (0.48) CA12CA14CA2TET2GAA
SCHEMBL2583703 0.78 CA12 (0.48) CA12CA14CA2TET2GAA
SCHEMBL25039078 0.77 CA12 (0.53) CA12CA14CA2TET2GAA
SCHEMBL22475391 0.76 CA12 (0.47) CA12CA14CA2TET2GAA
SCHEMBL15592453 0.76 CA12 (0.47) CA12CA14CA2TET2GAA
SCHEMBL4674334 0.76 CA12 (0.47) CA12CA14CA2TET2GAA
SCHEMBL10667453 0.76 CA12 (0.47) CA12CA14CA2TET2GAA
SCHEMBL22345253 0.74 CA12 (0.42) CA12CA14CA2TET2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11203586-B2 Iridinesulfonamide compound and use method thereof CHIA TAI TIANQING PHARMACEUTICAL GROUP CO., LTD. (CN) 2021-12-21 US disclosed
US-11203586-B2 Iridinesulfonamide compound and use method thereof CHIA TAI TIANQING PHARMACEUTICAL GROUP CO., LTD. (CN) 2021-12-21 US disclosed
US-11078168-B2 Substituted N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase Phenex Discovery Verwaltungs-GmbH (DE) 2021-08-03 US disclosed
US-20210155610-A1 Iridinesulfonamide Compound And Use Method Thereof LIANYUNGANG RUNZHONG PHARMACEUTICAL CO., LTD. (CN) 2021-05-27 US disclosed
US-20210155610-A1 Iridinesulfonamide Compound And Use Method Thereof LIANYUNGANG RUNZHONG PHARMACEUTICAL CO., LTD. (CN) 2021-05-27 US disclosed
CN-109071429-B Prophyridine sulfonamide compounds and methods of use thereof 正大天晴药业集团股份有限公司 2021-04-02 CN disclosed
EP-3444237-B1 IRIDINESULFONAMIDE COMPOUND AND USE METHOD THEREOF CHIA TAI TIANQING PHARMACEUTICAL GROUP CO LTD (CN) 2020-10-28 EP disclosed
EP-3444237-B1 IRIDINESULFONAMIDE COMPOUND AND USE METHOD THEREOF CHIA TAI TIANQING PHARMACEUTICAL GROUP CO LTD (CN) 2020-10-28 EP disclosed
US-20190292160-A1 SUBSTITUTED N-HYDROXYAMIDINOHETEROCYCLES AS MODULATORS OF INDOLEAMINE 2,3-DIOXYGENASE Phenex Discovery Verwaltungs-GmbH (DE) 2019-09-26 US disclosed
EP-3444237-A1 IRIDINESULFONAMIDE COMPOUND AND USE METHOD THEREOF Chai Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2019-02-20 EP disclosed
US-9073906-B2 Sulfamide derivative having an adamantyl group and its pharmaceutically acceptable salt KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2015-07-07 US disclosed
CN-104080766-A Sulphamide derivative having an adamantyl group and a pharmaceutically acceptable salt thereof KOREA RES INST CHEM TECH 2014-10-01 CN disclosed
EP-2740723-A2 SULPHAMIDE DERIVATIVE HAVING AN ADAMANTYL GROUP AND A PHARMACEUTICALLY ACCEPTABLE SALT THEREOF Korea Research Institute of Chemical Technology (KR) 2014-06-11 EP disclosed
US-20140024636-A1 SULFAMIDE DERIVATIVE HAVING AN ADAMANTYL GROUP AND ITS PHARMACEUTICALLY ACCEPTABLE SALT KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2014-01-23 US disclosed
US-20140024636-A1 SULFAMIDE DERIVATIVE HAVING AN ADAMANTYL GROUP AND ITS PHARMACEUTICALLY ACCEPTABLE SALT KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2014-01-23 US disclosed
EP-1137640-A1 CYCLIC HYDRAZINE DERIVATIVES AS TNF-ALPHA INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2001-10-04 EP disclosed
US-6281363-B1 ANTIINFLAMMATORY AGENTS; ANTIARTHRITIC AGENTS; AUTOIMMUNE DISORDERS HOFFMANN-LA ROCHE INC. 2001-08-28 US disclosed
WO-2000035885-A1 CYCLIC HYDRAZINE DERIVATIVES AS TNF-ALPHA INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2000-06-22 WO disclosed
US-5596017-A INSECTICIDES NIHON BAYER AGROCHEM K.K. (JP) 1997-01-21 US disclosed
EP-0684229-A1 Sulfamide derivatives NIHON BAYER AGROCHEM K.K. (JP) 1995-11-29 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11203586-B2 Iridinesulfonamide compound and use method thereof IDH1, IDH3B, IDH3A CA12 806/4885CA14 802/4885CA2 427/4885
US-11078168-B2 Substituted N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase IDO1, IDO2, INMT CA12 2596/4885CA14 3112/4885CA2 1506/4885
US-20140024636-A1 SULFAMIDE DERIVATIVE HAVING AN ADAMANTYL GROUP AND ITS PHARMACEUTICALLY ACCEPTABLE SALT HSD11B1, HSD11B2, HSD3B1 CA12 838/4885CA14 836/4885CA2 1279/4885
US-20210155610-A1 Iridinesulfonamide Compound And Use Method Thereof IDH1, IDH3B, IDH3A CA12 806/4885CA14 802/4885CA2 427/4885
US-20190292160-A1 SUBSTITUTED N-HYDROXYAMIDINOHETEROCYCLES AS MODULATORS OF INDOLEAMINE 2,3-DIOXYGENASE IDO1, IDO2, INMT CA12 2596/4885CA14 3112/4885CA2 1506/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.