SCHEMBL7841878

SCHEMBL7841878

CS(=O)(=O)c1ccc(NNc2cncc(Br)c2)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 1/20 0.40
PPARG P37231 5/20 0.39
SLC22A12 Q96S37 1/20 0.39
GCK P35557 2/20 0.37
CCR2 P41597 1/20 0.36
EPAS1 Q99814 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.35
EGFR P00533 1/20 0.34
CYP3A4 P08684 2/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
CA14 Q9ULX7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7841874 0.74 L3MBTL1 (0.44) GRM4PPARGGCKCCR2EPAS1
SCHEMBL12276475 0.72 CA1 (0.55) PPARGSLC22A12ALDH1A1CYP3A4CA1
SCHEMBL1581780 0.70 HSD11B1 (0.48) GRM4CCR2ALDH1A1CA1CA2
SCHEMBL29430629 0.70 HSD11B1 (0.48) GRM4CCR2ALDH1A1CA1CA2
SCHEMBL6534946 0.70 GRM4 (0.46) GRM4PPARGCCR2NPC1ALDH1A1
SCHEMBL22447441 0.69 SLC22A12 (0.55) PPARGSLC22A12CYP3A4CA1CA2
Hydrochloric Acid SCHEMBL6512600 0.68 GRM4 (0.45) GRM4PPARGCCR2NPC1ALDH1A1
SCHEMBL856308 0.68 PIK3CB (0.54) SLC22A12
SCHEMBL2312129 0.66 ALDH1A1 (0.69) SMN1; SMN2ALDH1A1
SCHEMBL12186139 0.65 L3MBTL1 (0.44) GRM4CCR2ALDH1A1CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1137647-A1 THIOUREA INHIBITORS OF HERPES VIRUSES AMERICAN HOME PRODUCTS CORPORATION (US) 2001-10-04 EP disclosed
WO-2000034268-A1 THIOUREA INHIBITORS OF HERPES VIRUSES AMERICAN HOME PRODUCTS CORPORATION (US) 2000-06-15 WO disclosed