SCHEMBL7842474

SCHEMBL7842474

O=C([CH]c1ccc(F)cc1)c1ccc(F)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNFRSF1A P19438 1/20 0.64
CES2 O00748 1/20 0.52
CES1 P23141 1/20 0.52
MAPT P10636 3/20 0.52
CYP1A1 P04798 1/20 0.51
CYP1B1 Q16678 1/20 0.51
CYP2C19 P33261 2/20 0.50
CYP1A2 P05177 1/20 0.50
MAOB P27338 2/20 0.49
MAOA P21397 1/20 0.49
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
HSD11B1 P28845 1/20 0.48
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
CTSL P07711 1/20 0.46
CTSB P07858 1/20 0.46
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2794365 0.90 TNFRSF1A (0.53) TNFRSF1ACES2CES1MAPTCYP1A1
SCHEMBL7448677 0.90 TNFRSF1A (0.53) TNFRSF1AMAPTCYP1B1CYP2C19CYP1A2
SCHEMBL8484185 0.86 LTA4H (0.58) TNFRSF1ACES2CES1MAPTCYP1A1
SCHEMBL6707524 0.86 LTA4H (0.58) TNFRSF1AMAPTCYP1A1CYP1B1CYP1A2
SCHEMBL7196521 0.78 TNFRSF1A (1.00) TNFRSF1AMAPTCYP1A1CYP1B1CYP2C19
SCHEMBL5593308 0.78 TNFRSF1A (1.00) TNFRSF1AMAPTCYP1A1CYP1B1CYP2C19
SCHEMBL6989990 0.78 TNFRSF1A (0.72) TNFRSF1ACES2CES1MAPTCYP1A1
SCHEMBL6989989 0.78 TNFRSF1A (0.72) TNFRSF1ACES2CES1MAPTCYP1A1
SCHEMBL4214525 0.76 TNFRSF1A (0.57) TNFRSF1ACES2CES1MAPTCYP1A1
SCHEMBL360314 0.76 MAPK1 (0.58) TNFRSF1ACES2CES1MAPTCYP1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1150565-A1 THIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF LION bioscience AG (DE) 2001-11-07 EP claimed
WO-2000045635-A1 THIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2000-08-10 WO claimed