SCHEMBL7448677

SCHEMBL7448677

O=C([CH]c1ccc(F)cc1)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNFRSF1A P19438 2/20 0.53
RAB9A P51151 3/20 0.53
NPC1 O15118 2/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
PLA2G7 Q13093 1/20 0.51
ALDH1A1 P00352 3/20 0.48
MAPK1 P28482 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
NFE2L2 Q16236 1/20 0.48
MAPT P10636 2/20 0.47
CYP3A4 P08684 2/20 0.47
PTGS2 P35354 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
KMT2A Q03164 2/20 0.47
MEN1 O00255 1/20 0.47
POLB P06746 1/20 0.47
MAOB P27338 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2794365 0.92 TNFRSF1A (0.53) TNFRSF1ARAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL7842474 0.90 TNFRSF1A (0.64) TNFRSF1ARAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL893710 0.85 CYP1B1 (0.61) TNFRSF1ARAB9AALDH1A1MAPK1TDP1
4-Fluoro Chalcone SCHEMBL657887 0.81 TNFRSF1A (0.82) TNFRSF1ARAB9AALDH1A1TDP1MAPT
4-Fluoro Chalcone SCHEMBL10363601 0.81 TNFRSF1A (0.82) TNFRSF1ARAB9AALDH1A1TDP1MAPT
SCHEMBL6707524 0.81 LTA4H (0.58) TNFRSF1ASMN1; SMN2MAPTPTGS2CYP1A2
4-Fluoro Chalcone SCHEMBL657888 0.81 TNFRSF1A (0.82) TNFRSF1ARAB9AALDH1A1TDP1MAPT
SCHEMBL4414022 0.80 MAPT (0.68) RAB9ANPC1SMN1; SMN2ALDH1A1MAPK1
SCHEMBL8484185 0.77 LTA4H (0.58) TNFRSF1ARAB9AMAPTPTGS2CYP1A2
SCHEMBL5950310 0.76 HSD11B1 (0.52) TNFRSF1ARAB9ANPC1SMN1; SMN2PLA2G7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6020347-A 4-substituted-4-piperidine carboxamide derivatives MERCK & CO., INC. (US) 2000-02-01 US disclosed
WO-1999025685-A1 4-SUBSTITUTED-4-PIPERIDINE CARBOXAMIDE DERIVATIVES MERCK & CO., INC. (US) 1999-05-27 WO disclosed