SCHEMBL7845199

SCHEMBL7845199

Cc1cc(C)cc(Sc2[nH]c(=O)n(Cc3ccccn3)c(=O)c2C(C)C)c1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 9/20 0.45
GRIN2B Q13224 9/20 0.45
NOX4 Q9NPH5 4/20 0.42
GABRA1 P14867 1/20 0.40
GABRA5 P31644 1/20 0.40
ALDH1A1 P00352 4/20 0.39
AGTR1 P30556 2/20 0.39
TLR7 Q9NYK1 1/20 0.39
KDM5B Q9UGL1 1/20 0.38
KDM4E B2RXH2 2/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7843371 0.85 ALDH1A1 (0.41) ALDH1A1TLR7KDM4EHPGD
SCHEMBL7845277 0.84 GRIN1 (0.45) GRIN1GRIN2BNOX4GABRA1GABRA5
SCHEMBL7848697 0.84 TLR7 (0.32) ALDH1A1TLR7KDM5BKDM4E
SCHEMBL6088087 0.84 GRIN1 (0.45) GRIN1GRIN2BNOX4GABRA1GABRA5
SCHEMBL7847101 0.80 GRIN1 (0.45) GRIN1GRIN2BNOX4GABRA1GABRA5
SCHEMBL7837569 0.78 KMT2A (0.37) GABRA1GABRA5ALDH1A1
SCHEMBL7837651 0.77 MTNR1A (0.50) GRIN1GRIN2BALDH1A1KDM4EHPGD
SCHEMBL7848879 0.77 TYMS (0.35)
SCHEMBL7849648 0.77 GRIN1 (0.36) GRIN1GRIN2BALDH1A1
SCHEMBL7848132 0.76 GRIN1 (0.40) GRIN1GRIN2BKDM5B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100786-A1 ANTIVIRAL PYRIMIDINEDIONE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF Samjin Pharmaceutical Co., Ltd. (KR) 2001-05-23 EP disclosed
WO-2000061564-A1 ANTIVIRAL PYRIMIDINEDIONE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF SAMJIN PHARMACEUTICAL CO., LTD. (KR) 2000-10-19 WO disclosed