SCHEMBL7849283

SCHEMBL7849283

CCS(=O)(=O)N(CC(=O)N(C)C)c1[c]cccc1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
ESR1 P03372 2/20 0.35
POLB P06746 2/20 0.35
NR4A1 P22736 1/20 0.35
OPRM1 P35372 1/20 0.34
OPRL1 P41146 1/20 0.34
HCRTR2 O43614 3/20 0.32
SMN1; SMN2 Q16637 2/20 0.31
NPSR1 Q6W5P4 1/20 0.31
KCNE1 P15382 1/20 0.31
KCNQ1 P51787 1/20 0.31
GRM2 Q14416 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2540120 0.80 ESR1 (0.35) ALDH1A1ESR1SMN1; SMN2GRM2
SCHEMBL7849438 0.75 ESR1 (0.33) ALDH1A1ESR1
SCHEMBL2536094 0.75 KCNE1 (0.33) ALDH1A1ESR1KCNE1KCNQ1
SCHEMBL7849449 0.75 SMN1; SMN2 (0.51) ALDH1A1POLBSMN1; SMN2
SCHEMBL7849862 0.75 OPRM1 (0.36) ALDH1A1NR4A1OPRM1OPRL1SMN1; SMN2
SCHEMBL7839475 0.74 KEAP1 (0.39) ALDH1A1POLBSMN1; SMN2
SCHEMBL2537926 0.73 ESR1 (0.33) ESR1
SCHEMBL2537879 0.70 NPC1 (0.33) ALDH1A1OPRM1SMN1; SMN2
SCHEMBL7839570 0.69 KDM4E (0.38) ALDH1A1ESR1POLBNR4A1
SCHEMBL11324580 0.69 TP53 (0.38) ALDH1A1ESR1SMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1115704-A1 NOVEL SUBSTITUTED INDOLINONES WITH AN INHIBITORY EFFECT ON VARIOUS KINASES AND CYCLIN/CDK COMPLEXES Boehringer Ingelheim Pharma KG (DE) 2001-07-18 EP disclosed
WO-2000018734-A1 NOVEL SUBSTITUTED INDOLINONES WITH AN INHIBITORY EFFECT ON VARIOUS KINASES AND CYCLIN/CDK COMPLEXES BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-04-06 WO disclosed