SCHEMBL7852010

SCHEMBL7852010

c1ccc(C2=NC(c3cccnc3)CC2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.44
CHRNA4 P43681 3/20 0.44
CYP11B2 P19099 2/20 0.44
CYP2A6 P11509 2/20 0.44
MAPK1 P28482 2/20 0.42
MAPT P10636 1/20 0.42
HTT P42858 1/20 0.42
CYP19A1 P11511 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
CHRNA7 P36544 2/20 0.41
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
CYP2D6 P10635 2/20 0.40
CYP2C19 P33261 2/20 0.40
POLB P06746 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
KDM4E B2RXH2 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5889312 0.85 NOS1 (0.49) MAPK1MAPTGAAMEN1KMT2A
SCHEMBL5889295 0.75 NOS1 (0.54) MAPTGAAMEN1KMT2AKDM4E
SCHEMBL14457906 0.74 ALDH1A1 (0.44) MAPK1MAPTALDH1A1MEN1KMT2A
SCHEMBL14457840 0.74 MAOA (0.47) MAPTALDH1A1GAAMEN1KMT2A
SCHEMBL14457932 0.74 NOS1 (0.42) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL24803124 0.72 CHRNB2 (0.58) CHRNB2CHRNA4CYP11B2CYP2A6ALDH1A1
SCHEMBL5889318 0.71 ALDH1A1 (0.56) MAPTALDH1A1GAAMEN1KMT2A
SCHEMBL14457874 0.71 CHRNB4 (0.45) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL4047125 0.70 IDO1 (0.39) CYP11B2CYP2A6ALDH1A1CYP2C19CYP1A2
SCHEMBL28699053 0.69 ALDH1A1 (0.49) CYP11B2CYP2A6MAPTHTTCYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1121357-A1 2-HETARYL-3,4-DIHYDRO-2H-PYRROLE DERIVATIVES Bayer Aktiengesellschaft (DE) 2001-08-08 EP disclosed
WO-2000021958-A1 2-HETARYL-3,4-DIHYDRO-2H-PYRROLE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2000-04-20 WO disclosed