SCHEMBL7854696

SCHEMBL7854696

CCCN1C(=O)C=CN(c2ccccc2)c2ccccc21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 7/20 0.37
GSK3A P49840 3/20 0.37
GSK3B P49841 3/20 0.37
MAPT P10636 2/20 0.36
ATM Q13315 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
LMNA P02545 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
ALDH1A1 P00352 3/20 0.35
HTT P42858 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
DRD2 P14416 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
PGR P06401 1/20 0.35
PTGS1 P23219 3/20 0.34
PTGS2 P35354 3/20 0.34
FAAH O00519 2/20 0.34
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7860353 0.74 ALDH1A1 (0.38) MAPTATMSMN1; SMN2LMNANPC1
SCHEMBL7854693 0.72 SMN1; SMN2 (0.37) MGLLGSK3AGSK3BMAPTSMN1; SMN2
SCHEMBL27345565 0.70 MGLL (0.52) MGLLGSK3AGSK3BATMNPC1
SCHEMBL16422227 0.70 LMNA (0.52) MAPTATMLMNAALDH1A1HTT
SCHEMBL15840870 0.68 GAA (0.41) MGLLGSK3AGSK3BATMLMNA
SCHEMBL7044712 0.67 HPGD (0.53) MAPTATMSMN1; SMN2LMNANPC1
SCHEMBL8083936 0.66 LMNA (0.46) MAPTLMNAALDH1A1HTTMEN1
SCHEMBL151770 0.66 MGLL (0.67) MGLLGSK3AGSK3BMAPTSMN1; SMN2
SCHEMBL7854683 0.65 BCHE (0.48) MAPTKMT2A
SCHEMBL7041976 0.65 CCKBR (0.50) SMN1; SMN2NPC1RAB9AALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0830350-B1 N-(1-ALKYL-5-PHENYL-2,3,4,5-TETRAHYDRO-1H-BENZO[B][1,5]DIAZEPIN-3-YL)-ACETAMIDES MERCK & CO INC (US) 2001-10-04 EP disclosed
US-5726171-A N-(1-alkyl-5-phenyl-2,3,4,5-tetrahydro-1H-benzo B! 1,4!diazepin-3yl)-acetamides MERCK & CO INC (US) 1998-03-10 US disclosed