4-Aminophenol

4-Aminophenol

SCHEMBL78547

Nc1ccc(O)cc1.O=P(O)(O)O

nearest known ligand 0.72

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of 4-Aminophenol. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.72
HIF1A Q16665 3/20 0.72
ALDH1A1 P00352 2/20 0.72
CA3 P07451 2/20 0.72
ALOX15 P16050 2/20 0.72
HSD17B10 Q99714 2/20 0.72
CA14 Q9ULX7 2/20 0.72
THRB P10828 2/20 0.72
CA6 P23280 1/20 0.72
CASP1 P29466 1/20 0.72
APP P05067 3/20 0.54
ESR1 P03372 3/20 0.46
CYP19A1 P11511 2/20 0.46
ESR2 Q92731 2/20 0.46
FDPS P14324 1/20 0.45
KDM4E B2RXH2 4/20 0.44
MAPT P10636 3/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
BLM P54132 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
4-Aminophenol SCHEMBL28849641 1.00 CYP3A4 (0.72) CYP3A4HIF1AALDH1A1CA3ALOX15
4-Aminophenol SCHEMBL28175334 0.97 CYP3A4 (0.68) CYP3A4HIF1AALDH1A1CA3ALOX15
Phosphoric Acid SCHEMBL6267680 0.88 MEN1 (0.57) CYP3A4HIF1AALDH1A1CA3ALOX15
4-Aminophenol SCHEMBL29019124 0.87 ALDH1A1 (0.54) CYP3A4HIF1AALDH1A1CA3ALOX15
4-Aminophenol SCHEMBL29019125 0.86 ALDH1A1 (0.77) CYP3A4HIF1AALDH1A1CA3ALOX15
Hydroquinone SCHEMBL329315 0.85 CA12 (0.61) CYP3A4HIF1AALDH1A1CA3ALOX15
Hydroquinone SCHEMBL131228 0.85 CA12 (0.61) CYP3A4HIF1AALDH1A1CA3ALOX15
4-Aminophenol SCHEMBL4861305 0.85 ALDH1A1 (1.00) CYP3A4HIF1AALDH1A1CA3ALOX15
4-Aminophenol SCHEMBL6753971 0.85 ALDH1A1 (1.00) CYP3A4HIF1AALDH1A1CA3ALOX15
4-Aminophenol SCHEMBL3424 0.85

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 708 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11919772-B2 Heteroatom doped polymer nanospheres/carbon nanospheres and preparation method thereof DALIAN UNIVERSITY OF TECHNOLOGY (CN) 2024-03-05 US claimed
US-20210253428-A1 Heteroatom doped Polymer Nanospheres/Carbon Nanospheres and Preparation Method Thereof DALIAN UNIVERSITY OF TECHNOLOGY (CN) 2021-08-19 US claimed
CN-108862240-B Heteroatom-doped carbon nano-microsphere and preparation method thereof 大连理工大学 2021-07-16 CN claimed
CN-109046191-B Core-shell structure nano material with hetero atom doped polymer as shell and preparation method thereof 大连理工大学 2021-04-23 CN claimed
CN-108822274-B Heteroatom-doped polymer nano-microsphere and preparation method thereof 大连理工大学 2021-03-19 CN claimed
CN-110711567-A Preparation method of high-performance nitrogen-containing porous carbon dioxide adsorbent 大连理工大学 2020-01-21 CN claimed
CN-109046191-A Core-shell structure nano material with hetero atom doped polymer as shell and preparation method thereof 大连理工大学 2018-12-21 CN claimed
CN-108862240-A Heteroatom-doped carbon nano-microsphere and preparation method thereof 大连理工大学 2018-11-23 CN claimed
CN-108822274-A Heteroatom-doped polymer nano-microsphere and preparation method thereof 大连理工大学 2018-11-16 CN claimed
WO-2013011513-A9 METHODS OF DETERMINING ENZYME ACTIVITY IN PRESERVED CELL SAMPLES RAMOT AT TEL-AVIV UNIVERSITY LTD. (IL) 2013-03-07 WO claimed
EP-1481246-B1 APPARATUS AND METHODS FOR ANALYTE MEASUREMENT AND IMMUNOASSAY I STAT CORP (US) 2008-09-10 EP claimed
US-7419821-B2 Apparatus and methods for analyte measurement and immunoassay I-STAT CORPORATION (US) 2008-09-02 US claimed
JP-2008525037-A 2008-07-17 JP claimed
EP-1871527-A2 MOLECULAR DIAGNOSTICS SYSTEM AND METHODS I-STAT CORPORATION (US) 2008-01-02 EP claimed
WO-2006071770-A2 MOLECULAR DIAGNOSTICS SYSTEM AND METHODS I-STAT CORPORATION (US) 2006-07-06 WO claimed
EP-1481246-A2 APPARATUS AND METHODS FOR ANALYTE MEASUREMENT AND IMMUNOASSAY I-STAT CORPORATION (US) 2004-12-01 EP claimed
WO-2003076937-A9 APPARATUS AND METHODS FOR ANALYTE MEASUREMENT AND IMMUNOASSAY I STAT CORP (US) 2004-04-22 WO claimed
WO-2003076937-A2 APPARATUS AND METHODS FOR ANALYTE MEASUREMENT AND IMMUNOASSAY I-STAT CORPORATION (US) 2003-09-18 WO claimed
US-20030170881-A1 Apparatus and methods for analyte measurement and immuno assay I-STAT CORPORATION 2003-09-11 US claimed
US-6391549-B1 DETECTING PARAMATER IN HOST CELL BY TRANSFECTING CELL WITH PLASMID WITH B-GALACTOSIDASE OR ALKALINE PHOSPHATASE REPORTER GENE UNDER CONTROL OF INDUCIBLE PROMOTER, ENZYMES CATALYZE REACTION CAUSING SIGNAL DETECTABLE BY ELECTROCHEMICAL CELL RAMONT UNIVERSITY AUTHORITY FOR APPLIED RESEARCH & INDUSTRIAL DEVELOPMENT LTD. (IL) 2002-05-21 US claimed