(2-Hydroxy-3-Imidazo[1,2-A]Pyridin-3-Yl-2-Phosphonopropionic Acid (Enantionmers)

(2-Hydroxy-3-Imidazo[1,2-A]Pyridin-3-Yl-2-Phosphonopropionic Acid (Enantionmers)

SCHEMBL7858749

O=C(O)C(O)(Cc1cnc2ccccn12)P(=O)(O)O

nearest known ligand 0.72

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FDPS P14324 3/20 0.72
GGPS1 O95749 1/20 0.72
GPR84 Q9NQS5 1/20 0.43
NPC1 O15118 6/20 0.40
RAB9A P51151 6/20 0.40
SMN1; SMN2 Q16637 5/20 0.40
ALDH1A1 P00352 5/20 0.40
HPGD P15428 4/20 0.40
KDM4E B2RXH2 2/20 0.40
GLA P06280 1/20 0.40
GAA P10253 1/20 0.40
ERCC5 P28715 1/20 0.40
NPSR1 Q6W5P4 2/20 0.39
EPHB3 P54753 1/20 0.38
HDAC1 Q13547 1/20 0.38
MAPT P10636 2/20 0.36
TP53 P04637 2/20 0.36
NAMPT P43490 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Minodronic Acid SCHEMBL145238 0.84 FDPS (1.00) FDPSGGPS1GPR84NPC1RAB9A
Minodronic Acid SCHEMBL6009958 0.83 FDPS (0.97) FDPSGGPS1GPR84NPC1RAB9A
Minodronic Acid SCHEMBL8661646 0.83 FDPS (0.97) FDPSGGPS1GPR84NPC1RAB9A
SCHEMBL23272074 0.81 FDPS (0.49) FDPSGGPS1LMNA
SCHEMBL12309035 0.80 FDPS (0.73) FDPSGGPS1GPR84NPC1RAB9A
Minodronic Acid SCHEMBL8661643 0.80 FDPS (0.85) FDPSGGPS1GPR84NPC1RAB9A
SCHEMBL17519343 0.80 FDPS (0.72) FDPSGGPS1GPR84NPC1RAB9A
SCHEMBL28033480 0.80 FDPS (0.72) FDPSGGPS1GPR84NPC1RAB9A
Minodronic Acid SCHEMBL8664061 0.79 FDPS (0.83) FDPSGGPS1GPR84NPC1RAB9A
Minodronic Acid SCHEMBL8659642 0.79 FDPS (0.83) FDPSGGPS1GPR84NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11400104-B2 Skeletal removal of bisphosphonates THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-08-02 US claimed
CN-109219438-B Bone removal of bisphosphonates 加州大学董事会 2022-04-22 CN claimed
US-20210121485-A1 Skeletal Removal of Bisphosphonates UNIV CALIFORNIA (US) 2021-04-29 US claimed
US-10857165-B2 Skeletal removal of bisphosphonates THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2020-12-08 US disclosed
US-20190209590-A1 Skeletal Removal of Bisphosphonates UNIVERSITY OF SOUTHERN CALIFORNIA 2019-07-11 US disclosed
EP-3463380-A1 SKELETAL REMOVAL OF BISPHOSPHONATES The Regents of The University of California (US) 2019-04-10 EP disclosed
US-20180064829-A1 FLUORESCENT BISPHOSPHONATE ANALOGS UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2018-03-08 US disclosed
EP-3278107-A1 FLUORESCENT BISPHOSPHONATE ANALOGS University of Southern California (US) 2018-02-07 EP disclosed
WO-2017210272-A1 SKELETAL REMOVAL OF BISPHOSPHONATES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2017-12-07 WO disclosed
WO-2016161407-A1 FLUORESCENT BISPHOSPHONATE ANALOGS UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2016-10-06 WO disclosed
EP-0788362-B1 PHOSPONOCARBOXYLATE COMPOUNDS FOR TREATING ABNORMAL CALCIUM AND PHOSPHATE METABOLISM PROCTER & GAMBLE PHARMA (US) 2001-07-25 EP disclosed
CN-1048017-C Phosphonocarboxylate compounds and pharmaceutical compositions containing the same PROCTER & GAMBLE PHARMA (US) 2000-01-05 CN disclosed
CN-1230409-A Phosphonocarboxylate compounds and pharmaceutical compositions containing the same PROCTER & GAMBLE PHARMA (US) 1999-10-06 CN disclosed
CN-1224018-A Phosphonic carboxylate compounds, pharmaceutical compositions contg. same PROCTER & GAMBLE PHARMA (US) 1999-07-28 CN disclosed
US-5760021-A TREATING OR PREVENTING METABOLIC BONE DISORDERS THE PROCTER & GAMBLE COMPANY (US) 1998-06-02 US disclosed
EP-0788362-A1 PHOSPONOCARBOXYLATE COMPOUNDS FOR TREATING ABNORMAL CALCIUM AND PHOSPHATE METABOLISM PROCTER & GAMBLE PHARMACEUTICALS, INC. (US) 1997-08-13 EP disclosed
CN-1089613-A Phosphonocarboxylate compounds and pharmaceutical compositions containing the same PROCTER & GAMBLE PHARMA (US) 1994-07-20 CN disclosed
WO-1993024131-A1 PHOSPONOCARBOXYLATE COMPOUNDS FOR TREATING ABNORMAL CALCIUM AND PHOSPHATE METABOLISM PROCTER & GAMBLE PHARMACEUTICALS, INC. (US) 1993-12-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210121485-A1 Skeletal Removal of Bisphosphonates SOST, ACP3, PTH1R FDPS 1272/4885GGPS1 271/4885GPR84 3461/4885
US-20180064829-A1 FLUORESCENT BISPHOSPHONATE ANALOGS PPIP5K2, PHPT1, PTH1R FDPS 362/4885GGPS1 215/4885GPR84 3637/4885
US-20190209590-A1 Skeletal Removal of Bisphosphonates SOST, ACP3, PTH1R FDPS 1272/4885GGPS1 271/4885GPR84 3461/4885
US-11400104-B2 Skeletal removal of bisphosphonates SOST, ACP3, PTH1R FDPS 1272/4885GGPS1 271/4885GPR84 3461/4885
US-10857165-B2 Skeletal removal of bisphosphonates SOST, ACP3, PTH1R FDPS 1272/4885GGPS1 271/4885GPR84 3461/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.