SCHEMBL7861165

SCHEMBL7861165

CS(=O)(=O)c1ccc(C(C=O)c2ccc(Br)cc2)cc1F

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 3/20 0.35
NMT1 P30419 1/20 0.33
AKR1B1 P15121 1/20 0.33
KCNH2 Q12809 1/20 0.32
PIK3CD O00329 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32
PIK3CG P48736 1/20 0.32
TBXA2R P21731 1/20 0.32
PTGDR Q13258 1/20 0.32
AKR1C3 P42330 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7863630 0.79 CCR2 (0.36) CCR2KCNH2PIK3CDPIK3CAPIK3CB
SCHEMBL29430705 0.76 NMT1 (0.49) CCR2NMT1AKR1B1CA1CA2
SCHEMBL1581645 0.76 NMT1 (0.49) CCR2NMT1AKR1B1CA1CA2
SCHEMBL11993144 0.73 CCR2 (0.41) CCR2KCNH2PIK3CDPIK3CAPIK3CB
SCHEMBL7861158 0.71 HDAC4 (0.42)
SCHEMBL6513419 0.70 ALDH1A1 (0.44) KCNH2PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL7448176 0.70 ALDH1A1 (0.44) KCNH2PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL21164275 0.69 CCR2 (0.38) CCR2KCNH2PIK3CDPIK3CAPIK3CB
SCHEMBL26999435 0.69 ALDH1A1 (0.54)
SCHEMBL48662 0.69 PIK3CD (0.39) CCR2KCNH2PIK3CDPIK3CAPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1086097-A1 SULFONYLBENZENE COMPOUNDS AS ANTI-INFLAMMATORY/ANALGESIC AGENTS PFIZER INC. (US) 2001-03-28 EP disclosed
WO-1999064415-A1 SULFONYLBENZENE COMPOUNDS AS ANTI-INFLAMMATORY/ANALGESIC AGENTS PFIZER PHARMACEUTICALS INC. (JP) 1999-12-16 WO disclosed