SCHEMBL7861390

SCHEMBL7861390

[C-]#[N+]CCc1ccc(O)cc1.c1ccc(COCc2ccccc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.50
LMNA P02545 2/20 0.44
CYP1A2 P05177 1/20 0.44
PTGS1 P23219 1/20 0.44
SLC6A2 P23975 1/20 0.44
CYP2C19 P33261 1/20 0.44
PTGS2 P35354 1/20 0.44
SLC6A3 Q01959 1/20 0.44
HIF1A Q16665 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
BCHE P06276 2/20 0.42
ESR1 P03372 2/20 0.42
ESR2 Q92731 2/20 0.42
FNTA P49354 1/20 0.41
FNTB P49356 1/20 0.41
KDM4E B2RXH2 1/20 0.40
POLB P06746 1/20 0.40
SLC2A1 P11166 1/20 0.40
IDO1 P14902 1/20 0.40
OPRM1 P35372 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7859899 0.84 ESR1 (0.59) LMNAPTGS1SLC6A2CYP2C19PTGS2
SCHEMBL1840533 0.82 TSHR (0.75) TSHRLMNACYP1A2PTGS1SLC6A2
SCHEMBL1461571 0.80 ALDH1A1 (0.48) TSHRLMNACYP1A2PTGS1SLC6A2
Hydroquinone SCHEMBL51561 0.80 TSHR (0.79) TSHRLMNACYP1A2PTGS1SLC6A2
SCHEMBL7861391 0.78 LTA4H (0.58) LMNACYP1A2PTGS1SLC6A2CYP2C19
Hydroquinone SCHEMBL7511716 0.78 TSHR (0.75) TSHRLMNACYP1A2PTGS1SLC6A2
SCHEMBL1837574 0.77 ESR1 (0.54) TSHRLMNACYP1A2PTGS1SLC6A2
SCHEMBL6744772 0.77 ESR1 (0.54) TSHRLMNACYP1A2PTGS1SLC6A2
Phenol SCHEMBL5486172 0.75 TSHR (0.79) TSHRLMNACYP1A2PTGS1SLC6A2
Phenol SCHEMBL21518644 0.75 TSHR (0.79) TSHRLMNACYP1A2PTGS1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070084-A4 PIPERAZINES AS INHIBITORS OF FRUCTOSE-1,6-BISPHOSPHATASE (FBPase) ONTOGEN CORP (US) 2001-09-12 EP disclosed
EP-1070084-A1 PIPERAZINES AS INHIBITORS OF FRUCTOSE-1,6-BISPHOSPHATASE (FBPase) Ontogen Corporation (US) 2001-01-24 EP disclosed
US-6107274-A ENZYME INHIBITORS AS HYPOGLYCEMIC AGENTS IN TREATMENT OF TYPE-II DIABETES ONTOGEN CORPORATION (US) 2000-08-22 US disclosed
WO-1999047549-A1 PIPERAZINES AS INHIBITORS OF FRUCTOSE-1,6-BISPHOSPHATASE (FBPase) ONTOGEN CORPORATION (US) 1999-09-23 WO disclosed