SCHEMBL7861969

SCHEMBL7861969

O=C(O)CC(c1ccccc1)c1cccc(CNC(=O)c2cccc(NC(=O)NCc3ccccc3)c2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.52
LMNA P02545 2/20 0.52
ITGB3 P05106 1/20 0.52
ITGAV P06756 1/20 0.52
CASR P41180 2/20 0.51
ALDH1A1 P00352 2/20 0.50
HPGD P15428 1/20 0.50
HTT P42858 1/20 0.50
KDR P35968 1/20 0.49
PPARG P37231 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC8 Q9BY41 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.48
SENP1 Q9P0U3 2/20 0.48
RAB9A P51151 2/20 0.48
NPC1 O15118 1/20 0.48
MITF O75030 1/20 0.48
KMT2A Q03164 1/20 0.48
SIRT2 Q8IXJ6 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7863288 0.87 SIRT2 (0.48) MAPK1LMNAITGB3ALDH1A1HPGD
SCHEMBL7861966 0.87 NAMPT (0.55) MAPK1LMNACASRALDH1A1HPGD
SCHEMBL7862052 0.83 MAPK1 (0.52) MAPK1LMNACASRALDH1A1HPGD
SCHEMBL7864712 0.82 SIRT2 (0.45) MAPK1LMNAITGB3ITGAVALDH1A1
SCHEMBL6778398 0.81 ITGB3 (0.59) MAPK1LMNAITGB3ITGAVALDH1A1
SCHEMBL7856448 0.81 PPARG (0.68) MAPK1LMNAITGB3ALDH1A1HPGD
SCHEMBL7856421 0.81 LMNA (0.44) MAPK1LMNAALDH1A1HPGDHTT
SCHEMBL7856420 0.81 LMNA (0.44) MAPK1LMNAALDH1A1HPGDHTT
SCHEMBL2836293 0.80 MAPK1 (0.51) MAPK1LMNAITGB3ITGAVCASR
SCHEMBL7864274 0.79 LMNA (0.43) MAPK1LMNAITGB3ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed
EP-0889877-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1999-01-13 EP claimed
WO-1997036862-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP disclosed
EP-0889877-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1999-01-13 EP disclosed
WO-1997036862-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1997-10-09 WO disclosed