SCHEMBL7866946

SCHEMBL7866946

NN=CNc1cccc(CCc2cccc(CC(C(=O)O)c3ccccc3)c2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.41
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39
FFAR1 O14842 2/20 0.38
CTSB P07858 4/20 0.37
SIRT1 Q96EB6 1/20 0.37
BACE1 P56817 1/20 0.36
BACE2 Q9Y5Z0 1/20 0.36
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36
MMP2 P08253 1/20 0.36
MMP3 P08254 1/20 0.36
CTSL P07711 1/20 0.35
CTSS P25774 1/20 0.35
CYP2C19 P33261 1/20 0.35
FNTA P49354 1/20 0.35
FNTB P49356 1/20 0.35
PGGT1B P53609 1/20 0.35
P4HTM Q9NXG6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7862057 0.88 ALDH1A1 (0.41) EPHX1FFAR1CTSB
SCHEMBL7864788 0.84 SIRT2 (0.44)
SCHEMBL7864160 0.81 FFAR1 (0.39) FFAR1SIRT1ITGB3ITGA2BCYP2C19
SCHEMBL7378809 0.80 NR1H4 (0.50) FFAR1ITGB3ITGA2B
SCHEMBL30902537 0.79 NOS3 (0.60) NOS3NOS1NOS2
SCHEMBL8075755 0.76 NOS3 (0.43) NOS3NOS1NOS2MMP2
SCHEMBL7864170 0.74 EPHX2 (0.47)
SCHEMBL7856489 0.74 ITGB3 (0.55) FFAR1SIRT1ITGB3ITGA2BMMP2
SCHEMBL7866927 0.72 FFAR1 (0.45) FFAR1ITGB3
SCHEMBL27501985 0.71 ITGB1 (0.44) ITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed