SCHEMBL7863151

SCHEMBL7863151

N=C(N)Nc1cccc(COc2cccc(C(CC(=O)O)c3ccccc3)c2)c1

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
FFAR1 O14842 2/20 0.47
F7 P08709 1/20 0.47
CTSA P10619 1/20 0.46
NR1H4 Q96RI1 1/20 0.46
SIRT2 Q8IXJ6 4/20 0.45
SIRT3 Q9NTG7 3/20 0.45
LTA4H P09960 3/20 0.45
SIRT1 Q96EB6 2/20 0.45
F10 P00742 1/20 0.44
MEN1 O00255 1/20 0.44
SGMS2 Q8NHU3 1/20 0.44
PDK1 Q15118 1/20 0.43
PDK2 Q15119 1/20 0.43
PDK3 Q15120 1/20 0.43
PDK4 Q16654 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7195712 0.85 ITGB3 (0.51) KMT2ASMN1; SMN2F7LTA4H
SCHEMBL7863285 0.84 ITGB3 (0.48) SIRT1F10
SCHEMBL7863159 0.84 KMT2A (0.56) KMT2ASMN1; SMN2FFAR1CTSANR1H4
SCHEMBL7863273 0.81 FFAR1 (0.43) FFAR1
SCHEMBL4028152 0.80 MAPK1 (0.58) KMT2ANR1H4SIRT2LTA4HF10
SCHEMBL7864754 0.79 PTPN11 (0.48) FFAR1
SCHEMBL7188076 0.79 F2 (0.44) KMT2ASMN1; SMN2F7LTA4HF10
SCHEMBL3910191 0.78 KMT2A (0.67) KMT2ASMN1; SMN2CTSASIRT2
SCHEMBL7864761 0.77 ITGB3 (0.43) KMT2AMEN1
SCHEMBL7856431 0.77 HDAC1 (0.45) KMT2ASMN1; SMN2SIRT1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP disclosed
EP-0889877-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1999-01-13 EP disclosed
WO-1997036862-A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS G.D. SEARLE & CO. (US) 1997-10-09 WO disclosed