SCHEMBL7863285

SCHEMBL7863285

N=C(N)Nc1cccc(CCc2cccc(C(CC(=O)O)c3ccccc3)c2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 4/20 0.48
ITGA2B P08514 3/20 0.48
SIRT1 Q96EB6 1/20 0.41
MAPT P10636 2/20 0.41
GAA P10253 1/20 0.41
LMNA P02545 1/20 0.40
AOC3 Q16853 1/20 0.40
F10 P00742 2/20 0.40
POLB P06746 1/20 0.40
MAPK1 P28482 1/20 0.40
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39
TPSAB1 Q15661 1/20 0.38
TPSD1 Q9BZJ3 1/20 0.38
TPSG1 Q9NRR2 1/20 0.38
PARP1 P09874 1/20 0.38
PARP10 Q53GL7 1/20 0.38
ITGAV P06756 1/20 0.38
F2 P00734 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8501220 0.88 ITGB3 (0.42) ITGB3ITGA2BSIRT1POLBITGAV
SCHEMBL7863273 0.87 FFAR1 (0.43) ITGB3ITGA2BMAPTLMNAPOLB
SCHEMBL7862054 0.86 F10 (0.52) ITGB3ITGA2BMAPTGAALMNA
SCHEMBL7864761 0.84 ITGB3 (0.43) ITGB3ITGA2BMAPTPOLBITGAV
SCHEMBL7863151 0.84 KMT2A (0.57) SIRT1F10
SCHEMBL7863288 0.83 SIRT2 (0.48) ITGB3ITGA2BMAPTLMNAMAPK1
SCHEMBL7856539 0.83 ITGB3 (0.41) ITGB3MAPTLMNAITGAVALDH1A1
SCHEMBL7861978 0.82 ITGB3 (0.35) ITGB3ITGA2BMAPTGAALMNA
SCHEMBL7864160 0.82 FFAR1 (0.39) ITGB3ITGA2BSIRT1LMNAITGAV
SCHEMBL7856431 0.82 HDAC1 (0.45) ITGB3ITGA2BSIRT1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP disclosed