SCHEMBL8324841

SCHEMBL8324841

CCCCCC1C(C(=O)O)=C(C)NC(c2cccc(-n3ccnc3)c2)=C1C(=O)OCC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 7/20 0.46
TRPV1 Q8NER1 3/20 0.46
ALDH1A1 P00352 6/20 0.39
LMNA P02545 3/20 0.39
ALOX12 P18054 1/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CACNA1C Q13936 1/20 0.39
MAPT P10636 3/20 0.38
TP53 P04637 2/20 0.38
TMIGD3 P0DMS9 2/20 0.38
ADH5 P11766 1/20 0.38
MAPK1 P28482 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8325950 0.90 ADORA3 (0.46) ADORA3TRPV1ALDH1A1LMNAHTT
SCHEMBL7864235 0.85 ADORA3 (0.38) ADORA3TRPV1NPSR1CACNA1CMAPT
SCHEMBL8327248 0.81 ADORA3 (0.68) ADORA3TRPV1ALDH1A1LMNATP53
SCHEMBL8323854 0.80 ADORA3 (0.62) ADORA3ALDH1A1LMNAALOX12HTT
SCHEMBL8323850 0.80 ADORA3 (0.62) ADORA3ALDH1A1LMNAALOX12HTT
SCHEMBL8327558 0.80 ADORA3 (0.54) ADORA3TRPV1ALDH1A1LMNANPSR1
SCHEMBL7869546 0.76 ADORA3 (0.41) ADORA3TRPV1ALDH1A1LMNAALOX12
SCHEMBL30357940 0.73 CACNA1F (0.54) ADORA3ALDH1A1LMNACACNA1CMAPT
SCHEMBL7269131 0.73 CACNA1F (0.54) ADORA3ALDH1A1LMNACACNA1CMAPT
SCHEMBL8330375 0.72 ADORA3 (0.42) ADORA3TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0943615-A1 1,4-DIHYDROPYRIDINE DERIVATIVES Nikken Chemicals Company, Limited (JP) 1999-09-22 EP disclosed