SCHEMBL7864284

SCHEMBL7864284

CC(C)(C)OC(=O)C(Cc1ccccc1)c1cccc(NS(=O)(=O)c2cccc(NC(=O)NCc3ccccc3)c2)c1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 10/20 0.50
ITGB3 P05106 3/20 0.49
ITGAV P06756 3/20 0.49
GHSR Q92847 1/20 0.47
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
IDH1 O75874 2/20 0.43
MAPT P10636 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41
MAPK1 P28482 1/20 0.41
KMT2A Q03164 1/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7864224 0.96 NAMPT (0.51) NAMPTITGB3ITGAVGHSRCA12
SCHEMBL7856493 0.85 NAMPT (0.53) NAMPTITGB3ITGAVGHSRMAPT
SCHEMBL7861846 0.85 CA1 (0.44) GHSRCA12CA1CA2CA9
SCHEMBL7861976 0.83 CA12 (0.43) GHSRCA12CA1CA2CA9
SCHEMBL7864272 0.82 NAMPT (0.58) NAMPTITGB3ITGAVGHSRCA12
SCHEMBL7864723 0.81 TGFBR1 (0.38) NAMPTCA12CA1CA2CA9
SCHEMBL7856514 0.79 ITGB3 (0.64) NAMPTITGB3ITGAVGHSRCA12
SCHEMBL7864643 0.78 ALDH1A1 (0.39) GHSRCA12CA1CA2CA9
SCHEMBL7863252 0.74 ITGB3 (0.58) NAMPTITGB3ITGAVGHSRCA12
SCHEMBL20671545 0.73 CA12 (0.55) GHSRCA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed