SCHEMBL7861976

SCHEMBL7861976

CC(C)(C)OC(=O)C(Cc1cccc(NS(=O)(=O)c2cccc(NC(N)=S)c2)c1)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
ALDH1A1 P00352 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
HTR6 P50406 6/20 0.42
TGFBR1 P36897 1/20 0.42
PTGES O14684 1/20 0.40
LMNA P02545 2/20 0.40
MAPT P10636 2/20 0.40
MEN1 O00255 1/20 0.40
MAPK1 P28482 1/20 0.40
KMT2A Q03164 1/20 0.40
IDH1 O75874 4/20 0.40
PKM P14618 1/20 0.38
IKBKB O14920 1/20 0.38
GHSR Q92847 1/20 0.38
ST14 Q9Y5Y6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7861846 0.93 CA1 (0.44) CA12CA1CA2CA9ALDH1A1
SCHEMBL7864224 0.88 NAMPT (0.51) CA12CA1CA2CA9ALDH1A1
SCHEMBL7863294 0.87 HTR6 (0.48) CA12CA1CA2CA9ALDH1A1
SCHEMBL7864284 0.83 NAMPT (0.50) CA12CA1CA2CA9LMNA
SCHEMBL7864643 0.82 ALDH1A1 (0.39) CA12CA1CA2CA9ALDH1A1
SCHEMBL7861972 0.81 TGFBR1 (0.43) CA1CA2ALDH1A1TGFBR1LMNA
SCHEMBL7856532 0.79 CA1 (0.51) CA12CA1CA2CA9ALDH1A1
SCHEMBL7864723 0.77 TGFBR1 (0.38) CA12CA1CA2CA9ALDH1A1
SCHEMBL7856443 0.76 LMNA (0.45) ALDH1A1LMNAMAPTMEN1KMT2A
SCHEMBL7863291 0.74 ITGB3 (0.45) CA1CA2CA9HTR6MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP disclosed