SCHEMBL7865053

SCHEMBL7865053

NC(=O)C1=CN(C(c2ccccc2)c2ccccc2)C=CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 1/20 0.40
NPSR1 Q6W5P4 5/20 0.36
CRHBP P24387 1/20 0.36
CRHR2 Q13324 1/20 0.36
KMT2A Q03164 3/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
PKM P14618 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MAOB P27338 1/20 0.35
MAPT P10636 2/20 0.34
KDM4E B2RXH2 1/20 0.34
HPGD P15428 1/20 0.34
GAA P10253 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRK1 P41145 1/20 0.34
OPRL1 P41146 1/20 0.34
LMNA P02545 2/20 0.33
MEN1 O00255 1/20 0.33
CACNA1H O95180 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17313343 0.85 CYP2D6 (0.33) OPRD1NPSR1CYP1A2CYP2D6PKM
SCHEMBL20829870 0.76 LDHA (0.34)
SCHEMBL21753524 0.73 ALDH1A1 (0.38) NPSR1KMT2ACYP1A2CYP2D6PKM
SCHEMBL2205423 0.70 ADRA1D (0.41) KMT2AGAA
Hydrochloric Acid SCHEMBL3803201 0.69 ADRA1D (0.40) KMT2AGAA
SCHEMBL298933 0.68 RAB9A (0.40) KMT2ASMN1; SMN2MAPTKDM4EHPGD
SCHEMBL21753516 0.67 TSHR (0.40) NPSR1KMT2ACYP1A2SMN1; SMN2MAPT
SCHEMBL1274356 0.66 LDHA (0.36)
SCHEMBL7865094 0.66 LDHA (0.34) MAPTALDH1A1
SCHEMBL9425743 0.66 LDHA (0.34) LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE37449-E1 INCLUDING 1,4-REDUCTION OF DIMERIC IMINIUM INTERMEDIATE TO AN ENAMINE BY REACTION WITH A 1,4-DIHYDROPYRIDINE; OXIDATIVE TRANSFORMATION OF THE PRODUCT TO A SECOND IMINIUM INTERMEDIATE; REDUCTION OF THE SECOND INTERMEDIATE UNIVERSITY OF BRITISH COLUMBIA (CA) 2001-11-13 US disclosed
CN-1027266-C Process for synthesis of dimer alkaloid compounds UNIV BRITISH COLUMBIA (CA) 1995-01-04 CN disclosed
US-5047528-A Antiviral, Antitumor And Antileukemic Agents UNIVERSITY OF BRISTISH COLUMBIA (CA) 1991-09-10 US disclosed
CN-1034728-A The synthetic method of dimer alkaloid compounds UNIV BRITISH COLUMBIA (CA) 1989-08-16 CN disclosed