SCHEMBL7866465

SCHEMBL7866465

O=S(=O)(c1ccccc1)n1c(N2CCC(O)CC2)cc2ccccc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.45
CA12 O43570 3/20 0.44
CA9 Q16790 3/20 0.44
CA2 P00918 1/20 0.44
ALDH1A1 P00352 2/20 0.44
LMNA P02545 2/20 0.44
RECQL P46063 1/20 0.44
MAPT P10636 1/20 0.44
ALOX5 P09917 1/20 0.41
CCR2 P41597 1/20 0.40
SRC P12931 1/20 0.40
HDAC3 O15379 2/20 0.39
HDAC4 P56524 2/20 0.39
HDAC1 Q13547 2/20 0.39
HDAC7 Q8WUI4 2/20 0.39
HDAC2 Q92769 2/20 0.39
HDAC10 Q969S8 2/20 0.39
HDAC11 Q96DB2 2/20 0.39
HDAC8 Q9BY41 2/20 0.39
HDAC6 Q9UBN7 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4304442 0.82 HTR6 (0.54) CA12CA9CA2HTR6
Hydrochloric Acid SCHEMBL4316251 0.81 HTR6 (0.53) CA12CA9CA2HTR6
Hydrochloric Acid SCHEMBL6521806 0.81 HTR6 (0.53) CA12CA9CA2HTR6
SCHEMBL7085731 0.78 HTR6 (0.53) ALDH1A1LMNAHTR6TSHRKMT2A
SCHEMBL17422147 0.72 ALOX5 (0.52) ALDH1A1LMNAALOX5HTR6HPGD
SCHEMBL4316005 0.72 MAPT (0.51) ALDH1A1MAPTCCR2HTR6HPGD
SCHEMBL4309788 0.72 PKM (0.45) CA12CA9CA2LMNAMAPT
SCHEMBL4315943 0.72 LTA4H (0.48) CA12CA9CA2ALDH1A1LMNA
Hydrochloric Acid SCHEMBL6518308 0.72 HTR6 (0.44) CA12CA9CA2LMNAMAPT
Hydrochloric Acid SCHEMBL6518351 0.72 HTR6 (0.50) ALDH1A1MAPTCCR2HTR6HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077213-A2 Inhibition of serotonin reuptake ELI LILLY AND COMPANY (US) 2001-02-21 EP disclosed
US-6046215-A A PIPERIDINYLBENZOTHIOPHENES USEFUL FOR TRATING BRAIN DISORDERS ELI LILLY AND COMPANY (US) 2000-04-04 US disclosed
US-5846982-A Inhibition of serotonin reuptake ELI LILLY AND COMPANY (US) 1998-12-08 US disclosed
WO-1997047302-A1 INHIBITION OF SEROTONIN REUPTAKE ELI LILLY AND COMPANY (US) 1997-12-18 WO disclosed
EP-0812826-A1 1H-indole and benzo(b)thiophene derivatives with 4-(1,2,3,6-tetra:hydro:pyridinyl)- and 4-piperidinyl-groups bound to the heterocyclic ring as inhibitors of serotonin reuptake ELI LILLY AND COMPANY (US) 1997-12-17 EP disclosed