SCHEMBL7867464

SCHEMBL7867464

COc1ccc([CH]C#N)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.57
KDM4E B2RXH2 4/20 0.57
CYP1A2 P05177 4/20 0.57
CYP3A4 P08684 3/20 0.57
MAPT P10636 3/20 0.57
HPGD P15428 3/20 0.57
TSHR P16473 2/20 0.57
NFKB1 P19838 1/20 0.57
APEX1 P27695 1/20 0.57
BLM P54132 1/20 0.57
PMP22 Q01453 1/20 0.57
NPSR1 Q6W5P4 1/20 0.57
CYP2A6 P11509 1/20 0.52
LMNA P02545 1/20 0.50
TP53 P04637 1/20 0.50
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA7 P43166 1/20 0.50
CA9 Q16790 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2719499 0.82 NQO1 (0.49) ALDH1A1KDM4ECYP1A2CYP3A4MAPT
SCHEMBL442274 0.78 KDM4E (0.57) ALDH1A1KDM4ECYP1A2CYP3A4MAPT
SCHEMBL442275 0.78 KDM4E (0.57) ALDH1A1KDM4ECYP1A2CYP3A4MAPT
SCHEMBL3223495 0.77 ALDH1A1 (0.52) ALDH1A1KDM4ECYP1A2CYP3A4MAPT
SCHEMBL10549379 0.77 NFE2L2 (0.42) ALDH1A1KDM4ECYP1A2CYP3A4MAPT
Acrylonitrile SCHEMBL10901156 0.77 ALDH1A1 (0.52) ALDH1A1KDM4ECYP1A2CYP3A4MAPT
SCHEMBL10545617 0.77 RELA (0.51) ALDH1A1KDM4ECYP1A2TRPA1RELA
SCHEMBL10975899 0.74 LTA4H (0.50) ALDH1A1HPGDTSHRLMNACA1
SCHEMBL6247331 0.74 KDM4E (0.53) ALDH1A1KDM4ECYP1A2CYP3A4MAPT
SCHEMBL6247325 0.74 KDM4E (0.53) ALDH1A1KDM4ECYP1A2CYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1086107-A1 ARTEMISININ DERIVATIVES, METHOD FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME SHANGHAI INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF SCIENCES (CN) 2001-03-28 EP disclosed
WO-1999065914-A1 ARTEMISININ DERIVATIVES, METHOD FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME SHANGHAI INSTITUTE OF MATERIA MEDICA (CN) 1999-12-23 WO disclosed