SCHEMBL7868005

SCHEMBL7868005

CCN1CC=C(c2[nH]c3cc(C#N)ccc3c2OC(=O)C(=O)Oc2c(C3=CCN(CC)CC3)[nH]c3cc(C#N)ccc23)CC1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.41
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.40
ALOX15 P16050 1/20 0.40
ALK Q9UM73 5/20 0.40
PARP1 P09874 2/20 0.38
SLC6A4 P31645 1/20 0.37
HTR1A P08908 2/20 0.37
CCNT1 O60563 1/20 0.36
CDK9 P50750 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7868031 0.93 HTR6 (0.46) HTR6KDM4ELMNAALOX15ALK
SCHEMBL7867413 0.82 KDM4E (0.39) HTR6KDM4ELMNAALOX15PARP1
SCHEMBL7866250 0.80 KDM4E (0.41) HTR6KDM4ELMNAALOX15CCNT1
SCHEMBL7867440 0.76 HRH3 (0.45) ALK
Oxalic Acid SCHEMBL7865005 0.74 KDM4E (0.59) HTR6KDM4ELMNAALOX15SLC6A4
Oxalic Acid SCHEMBL7867999 0.73 DRD2 (0.41) HTR6KDM4ELMNAALOX15PARP1
Oxalic Acid SCHEMBL7868026 0.73 CYP19A1 (0.44) HTR6ALKPARP1SLC6A4CCNT1
SCHEMBL7870827 0.72 KDM4E (0.37) HTR6KDM4ELMNAALOX15PARP1
Oxalic Acid SCHEMBL7867306 0.71 SLC6A4 (0.66) HTR6KDM4ELMNAALOX15SLC6A4
Oxalic Acid SCHEMBL7867561 0.69 HTR1D (0.40) KDM4ELMNAALOX15ALKPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077213-A2 Inhibition of serotonin reuptake ELI LILLY AND COMPANY (US) 2001-02-21 EP disclosed
US-6046215-A A PIPERIDINYLBENZOTHIOPHENES USEFUL FOR TRATING BRAIN DISORDERS ELI LILLY AND COMPANY (US) 2000-04-04 US disclosed
US-5846982-A Inhibition of serotonin reuptake ELI LILLY AND COMPANY (US) 1998-12-08 US disclosed
EP-0812826-A1 1H-indole and benzo(b)thiophene derivatives with 4-(1,2,3,6-tetra:hydro:pyridinyl)- and 4-piperidinyl-groups bound to the heterocyclic ring as inhibitors of serotonin reuptake ELI LILLY AND COMPANY (US) 1997-12-17 EP disclosed