SCHEMBL7868624

SCHEMBL7868624

CC(=O)c1ccc(-n2ccnc2)cc1.CON=C(C)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.58
BAZ2B Q9UIF8 1/20 0.58
MAPT P10636 8/20 0.50
LMNA P02545 4/20 0.50
HTT P42858 2/20 0.49
L3MBTL1 Q9Y468 2/20 0.47
ADH5 P11766 2/20 0.45
SMN1; SMN2 Q16637 3/20 0.43
RAB9A P51151 2/20 0.43
NPSR1 Q6W5P4 1/20 0.43
ALDH1A1 P00352 3/20 0.43
HPGD P15428 1/20 0.43
AHR P35869 1/20 0.41
NPC1 O15118 1/20 0.41
GAA P10253 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL611481 0.76 CYP3A4 (1.00) CYP3A4BAZ2BMAPTLMNAHTT
Trifluoromethanesulfonic Acid SCHEMBL5694136 0.76 CYP3A4 (0.76) CYP3A4BAZ2BMAPTLMNAHTT
SCHEMBL6819613 0.74 CES2 (0.45) MAPTNPSR1GAAMEN1KMT2A
SCHEMBL3535504 0.68 ADH5 (0.54) CYP3A4BAZ2BHTTADH5ALDH1A1
SCHEMBL1882019 0.68 CYP3A4 (0.47) CYP3A4MAPTLMNAADH5ALDH1A1
SCHEMBL709619 0.68 LMNA (0.58) CYP3A4BAZ2BMAPTLMNAHTT
SCHEMBL1022965 0.67 HTT (1.00) CYP3A4BAZ2BMAPTLMNAHTT
SCHEMBL8333311 0.67 CYP11B1 (0.55) CYP3A4MAPTLMNAHTTSMN1; SMN2
Hydrochloric Acid SCHEMBL17583800 0.67 CYP3A4 (0.46) CYP3A4MAPTLMNAADH5ALDH1A1
Benzaldehyde SCHEMBL27623570 0.66 CYP3A4 (0.76) CYP3A4BAZ2BMAPTLMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1137645-A2 ALPHA-METHYLBENZYL-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING A PHENYLENEDIAMINE GROUP AMERICAN HOME PRODUCTS CORPORATION (US) 2001-10-04 EP disclosed
WO-2000034260-A2 ALPHA-METHYLBENZYL-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING A PHENYLENEDIAMINE GROUP AMERICAN HOME PRODUCTS CORPORATION (US) 2000-06-15 WO disclosed