SCHEMBL7868830

SCHEMBL7868830

CC(CSc1ccc(OS(=O)(=O)C(F)(F)F)cc1)C(=O)OC(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 2/20 0.43
CXCR1 P25024 1/20 0.42
SDCBP O00560 1/20 0.36
SDC2 P34741 1/20 0.36
MMP2 P08253 1/20 0.35
ADAM17 P78536 1/20 0.35
PPARD Q03181 6/20 0.34
AAK1 Q2M2I8 1/20 0.34
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA4 P22748 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
HSD11B1 P28845 1/20 0.33
ALDH1A1 P00352 1/20 0.33
PPARA Q07869 1/20 0.32
MTNR1A P48039 3/20 0.32
MTNR1B P49286 3/20 0.32
DRD2 P14416 1/20 0.32
DRD1 P21728 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7867068 0.79 CXCR2 (0.43) CXCR2CXCR1MMP2ADAM17
SCHEMBL7862178 0.79 ADRB2 (0.38) SDCBPSDC2MMP2ADAM17CA1
SCHEMBL19890873 0.73 MTNR1A (0.43) AAK1CA1CA2CA4CA7
SCHEMBL4652349 0.71 CXCR2 (0.50) CXCR2CXCR1PPARDPPARA
SCHEMBL3843634 0.70 CA12 (0.51) CXCR2CXCR1CA1CA2CA9
SCHEMBL17195668 0.70 CA12 (0.50) CXCR2CXCR1SDCBPSDC2CA1
SCHEMBL7048726 0.70 LDHA (0.40) CXCR2CXCR1PPARDPPARA
SCHEMBL27620195 0.70 PTPN1 (0.41) CXCR2CXCR1PPARA
SCHEMBL2863819 0.69 KDM4E (0.43) CXCR2
SCHEMBL2856829 0.69 ITGB3 (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6300514-B1 INHIBITING MATRIX METALLOPROTEINASES ONO PHARMACEUTICAL CO., LTD. (JP) 2001-10-09 US disclosed
EP-0994104-A1 ARYL (SULFIDE, SULFOXIDE AND SULFONE) DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2000-04-19 EP disclosed