SCHEMBL7869050

SCHEMBL7869050

CCCCC(NCc1ccco1)c1ccc(C(=O)O)c(-c2ccccc2C)c1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP2C9 P11712 1/20 0.41
GAA P10253 4/20 0.41
ALDH1A1 P00352 3/20 0.41
PKM P14618 1/20 0.41
MAPT P10636 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TDP1 Q9NUW8 2/20 0.39
KDM4E B2RXH2 1/20 0.39
NPSR1 Q6W5P4 2/20 0.38
APP P05067 2/20 0.37
USP2 O75604 2/20 0.37
MAPK1 P28482 1/20 0.37
HPGD P15428 1/20 0.37
MEN1 O00255 1/20 0.37
HTT P42858 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7869068 0.81 ADRB1 (0.38) CYP1A2CYP2C19CYP2C9HPGD
SCHEMBL7871095 0.72 LTB4R2 (0.38) CYP1A2CYP2C19CYP2C9NPSR1HPGD
SCHEMBL7869054 0.71 FNTA (0.45) ALDH1A1MAPTL3MBTL1NPSR1
SCHEMBL7908229 0.70 PTPN11 (0.35)
SCHEMBL6625288 0.65 FNTA (0.42)
SCHEMBL4677601 0.64 TDP1 (0.50) CYP1A2CYP2C19CYP2C9GAAALDH1A1
SCHEMBL28552914 0.64 PLK1 (0.46)
SCHEMBL7918101 0.63 MYC (0.46) ALDH1A1KDM4EHPGDHTT
SCHEMBL29064695 0.62 MYC (0.56) GAAALDH1A1KDM4EUSP2HPGD
SCHEMBL7905474 0.62 SLC6A3 (0.38) ALDH1A1MAPTKDM4ENPSR1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6310095-B1 INHIBITING OR TREATING CANCER, TREATING INTIMAL HYPERPLASIA ASSOCIATED WITH RESTENOSIS AND ATHEROSCLEROSIS, INHIBITING POST-TRANSLATIONAL MODIFICATION OF ONCOGENIC RAS PROTEIN BY PROTEIN FARNESYLTRANSFERASE AND/OR GERANYLGERANYLTRANSFERASE UNIVERSITY OF PITTSBURGH 2001-10-30 US disclosed