SCHEMBL7869485

SCHEMBL7869485

CCCn1c(=O)[nH]c(=S)c2[nH]c(-c3ccc(Br)cc3)nc21

nearest known ligand 0.69

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 12/20 0.69
ADORA3 P0DMS8 1/20 0.64
ADORA2A P29274 7/20 0.60
ADORA1 P30542 1/20 0.53
KDM4E B2RXH2 1/20 0.52
MEN1 O00255 1/20 0.52
ALDH1A1 P00352 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
KMT2A Q03164 1/20 0.52
HSD17B10 Q99714 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7863965 0.90 ADORA2B (0.58) ADORA2BADORA3ADORA2AADORA1KDM4E
SCHEMBL7866628 0.89 ADORA2B (0.61) ADORA2BADORA3ADORA2AADORA1KDM4E
SCHEMBL7866612 0.88 ADORA2B (0.77) ADORA2BADORA3ADORA2AADORA1KDM4E
SCHEMBL7866293 0.81 ADORA2B (0.55) ADORA2BADORA2AADORA1KDM4EMEN1
SCHEMBL5229753 0.81 ADORA2B (0.55) ADORA2BADORA2AADORA1KDM4EMEN1
SCHEMBL7866617 0.78 ADORA2B (0.62) ADORA2BADORA3ADORA2AADORA1KDM4E
SCHEMBL5230505 0.77 ADORA2B (0.66) ADORA2BADORA3ADORA2AADORA1KDM4E
SCHEMBL7866286 0.77 ADORA2B (0.79) ADORA2BADORA3ADORA2AADORA1KDM4E
SCHEMBL9706669 0.75 ADORA2A (0.45) ADORA2BADORA3ADORA2AADORA1HSD17B10
SCHEMBL9765885 0.75 ADORA2B (1.00) ADORA2BADORA3ADORA2AADORA1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6306847-B1 ANTIALLERGENS AND BRONCHODILATOR AGENTS KYOWA HAKKO KOGYO CO., LTD. (JP) 2001-10-23 US disclosed
EP-0884318-A1 FUSED PURINE DERIVATIVES KYOWA HAKKO KOGYO CO., LTD. (JP) 1998-12-16 EP disclosed