SCHEMBL5229753

SCHEMBL5229753

CCCn1c(=O)[nH]c(=S)c2[nH]c(-c3ccsc3)nc21

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 8/20 0.55
ADORA2A P29274 5/20 0.55
ALDH1A1 P00352 2/20 0.53
HSD17B10 Q99714 2/20 0.53
KDM4A O75164 1/20 0.53
HPGD P15428 1/20 0.53
TSHR P16473 1/20 0.53
MAPK1 P28482 1/20 0.53
CASP1 P29466 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
KDM4C Q9H3R0 1/20 0.53
RXFP1 Q9HBX9 1/20 0.53
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
KMT2A Q03164 1/20 0.47
ADORA1 P30542 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7866628 0.82 ADORA2B (0.61) ADORA2BADORA2AALDH1A1HSD17B10KDM4E
SCHEMBL10675027 0.82 ADORA2B (0.70) ADORA2BADORA2AALDH1A1HSD17B10KDM4E
SCHEMBL7869485 0.81 ADORA2B (0.69) ADORA2BADORA2AALDH1A1HSD17B10KDM4E
SCHEMBL7866293 0.75 ADORA2B (0.55) ADORA2BADORA2AALDH1A1HSD17B10KDM4E
SCHEMBL9706669 0.73 ADORA2A (0.45) ADORA2BADORA2AHSD17B10HPGDADORA1
SCHEMBL7420292 0.72 ADORA1 (0.44) ADORA2BADORA2AHSD17B10HPGDADORA1
SCHEMBL7863965 0.71 ADORA2B (0.58) ADORA2BADORA2AALDH1A1HSD17B10HPGD
SCHEMBL9765885 0.71 ADORA2B (1.00) ADORA2BADORA2AALDH1A1HSD17B10HPGD
SCHEMBL7423540 0.70 ADORA2A (0.45) ADORA2BADORA2A
SCHEMBL5231243 0.70 PDE2A (0.46) ADORA2BADORA2AHSD17B10HPGDADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1092435-B1 REMEDIES FOR DIABETES KYOWA HAKKO KOGYO KK (JP) 2007-04-04 EP disclosed
US-6489331-B1 A CONDENSED PURINE DERIVATIVE AS AN ACTIVE INGREDIENT AS AN ENHANCER OF INSULIN SECRETION AND A MEDICAMENT FOR THE TREATMENT OF DIABETES KYOWA HAKKO KOGYO CO., LTD. (JP) 2002-12-03 US disclosed
EP-1092435-A1 REMEDIES FOR DIABETES KYOWA HAKKO KOGYO CO., LTD. (JP) 2001-04-18 EP disclosed