Arbutamine

Arbutamine

SCHEMBL7870502

O=C(O)C(=O)O.Oc1ccc(CCCCNC[C@H](O)c2ccc(O)c(O)c2)cc1

nearest known ligand 0.65

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

OPRM1SLC6A4

The experimentally established mechanism targets of Arbutamine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 known ✓ P31645 1/20 0.53
ADRB2 P07550 17/20 0.58
ADRB1 P08588 10/20 0.58
ADRB3 P13945 7/20 0.53
DRD2 P14416 3/20 0.53
DRD4 P21917 3/20 0.53
DRD3 P35462 3/20 0.53
ALOX15 P16050 2/20 0.53
KDM4E B2RXH2 1/20 0.53
HTR1A P08908 1/20 0.53
CHRM5 P08912 1/20 0.53
ADRA2B P18089 1/20 0.53
SLC6A2 P23975 1/20 0.53
FPR3 P25089 1/20 0.53
ADRA1D P25100 1/20 0.53
HTR1D P28221 1/20 0.53
HTR1B P28222 1/20 0.53
HTR2A P28223 1/20 0.53
HTR2C P28335 1/20 0.53
GPR183 P32249 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Arbutamine SCHEMBL29390265 0.94 ADRB2 (0.61) ADRB2ADRB1ADRB3DRD2DRD4
Arbutamine SCHEMBL20769823 0.94 ADRB2 (0.61) ADRB2ADRB1ADRB3DRD2DRD4
Arbutamine SCHEMBL521645 0.94 ADRB2 (0.61) ADRB2ADRB1ADRB3DRD2DRD4
Arbutamine SCHEMBL3699485 0.94 ADRB2 (0.61) ADRB2ADRB1ADRB3DRD2DRD4
Arbutamine SCHEMBL29929016 0.94 ADRB2 (0.61) ADRB2ADRB1ADRB3DRD2DRD4
Arbutamine SCHEMBL7295080 0.93 ADRB2 (0.60) ADRB2ADRB1ADRB3DRD2DRD4
Arbutamine SCHEMBL40757 0.93 ADRB2 (0.60) ADRB2ADRB1ADRB3DRD2DRD4
Arbutamine SCHEMBL4327619 0.91 ADRB2 (0.59) ADRB2ADRB1ADRB3DRD2DRD4
Arbutamine SCHEMBL8367936 0.88 ADRB2 (0.57) ADRB2ADRB1ADRB3DRD2DRD4
Oxalic Acid SCHEMBL11482348 0.86 SMN1; SMN2 (0.54) ADRB2ADRB1ADRB3KDM4ESLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0873293-B1 IMPROVED PROCESS FOR THE PREPARATION OF ALKYL OR ARYL ALDEHYDE INTERMEDIATES ABBOTT LAB (US) 2001-07-25 EP disclosed
EP-0873293-A1 IMPROVED PROCESS FOR THE PREPARATION OF ALKYL OR ARYL ALDEHYDE INTERMEDIATES Abbott Laboratories (US) 1998-10-28 EP disclosed
WO-1997023439-A1 IMPROVED PROCESS FOR THE PREPARATION OF ALKYL OR ARYL ALDEHYDE INTERMEDIATES ABBOTT LABORATORIES (US) 1997-07-03 WO disclosed