Arbutamine

Arbutamine

SCHEMBL521645

Oc1ccc(CCCCNC[C@H](O)c2ccc(O)c(O)c2)cc1

nearest known ligand 0.74

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 14/20 0.61
ADRB1 P08588 7/20 0.61
ADRB3 P13945 4/20 0.56
DRD2 P14416 4/20 0.55
DRD3 P35462 4/20 0.55
DRD4 P21917 3/20 0.55
MEN1 O00255 3/20 0.55
KMT2A Q03164 3/20 0.55
ALOX15 P16050 2/20 0.55
KDM4E B2RXH2 2/20 0.55
ADRA2B P18089 2/20 0.55
ADRA1D P25100 2/20 0.55
ADRA1A P35348 2/20 0.55
CYP1A2 P05177 2/20 0.55
CYP3A4 P08684 2/20 0.55
CYP2D6 P10635 2/20 0.55
TSHR P16473 2/20 0.55
MAPK1 P28482 2/20 0.55
HTR1A P08908 1/20 0.55
CHRM5 P08912 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Arbutamine SCHEMBL3699485 1.00 ADRB2 (0.61) ADRB2ADRB1ADRB3DRD2DRD3
Arbutamine SCHEMBL29929016 1.00 ADRB2 (0.61) ADRB2ADRB1ADRB3DRD2DRD3
Arbutamine SCHEMBL20769823 1.00 ADRB2 (0.61) ADRB2ADRB1ADRB3DRD2DRD3
Arbutamine SCHEMBL29390265 1.00 ADRB2 (0.61) ADRB2ADRB1ADRB3DRD2DRD3
Arbutamine SCHEMBL7295080 0.99 ADRB2 (0.60) ADRB2ADRB1ADRB3DRD2DRD3
Arbutamine SCHEMBL40757 0.99 ADRB2 (0.60) ADRB2ADRB1ADRB3DRD2DRD3
Arbutamine SCHEMBL4327619 0.97 ADRB2 (0.59) ADRB2ADRB1ADRB3DRD2DRD3
Arbutamine SCHEMBL7870502 0.94 ADRB2 (0.58) ADRB2ADRB1ADRB3DRD2DRD3
Hexoprenaline SCHEMBL121449 0.85 ADRB2 (0.72) ADRB2ADRB1ADRB3DRD2DRD3
Hexoprenaline SCHEMBL32668781 0.85 ADRB2 (0.72) ADRB2ADRB1ADRB3DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 952 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025265094-A1 COMPOSITIONS AND METHODS FOR TREATING METABOLIC DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2025-12-26 WO claimed
US-12485181-B2 Polyoxazoline-drug conjugates with novel pharmacokinetic properties SERINA THERAPEUTICS (AL), INC. (US) 2025-12-02 US claimed
US-12383625-B2 Polyoxazoline-drug conjugates with novel pharmacokinetic properties SERINA THERAPEUTICS (AL), INC. (US) 2025-08-12 US claimed
US-12383626-B2 Polyoxazoline-drug conjugates with novel pharmacokinetic properties SERINA THERAPEUTICS (AL), INC. (US) 2025-08-12 US claimed
US-20250213647-A1 CHEMOKINE RECEPTORS AND ALPHA1 ADRENERGIC RECEPTORS/VASOPRESSIN RECEPTORS 1A HETEROMERS AS DRUG TARGETS FOR DISEASE UNIVERSITY OF SOUTH FLORIDA 2025-07-03 US claimed
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO claimed
EP-4483376-A1 MEASUREMENT, DIAGNOSIS, TREATMENT AND MANAGEMENT OF METABOLIC SYNDROME García Sada, Fernando (MX) 2025-01-01 EP claimed
US-20240398729-A1 Methods and Compositions for the Treatment of Cytoplasmic Glycogen Storage Disorders DUKE UNIVERSITY (US) 2024-12-05 US claimed
US-20240390364-A1 Novel Pyridine Compositions and their use in methods for preventing or treating diseases, disorders and conditions REID CHRISTOPHER BRIAN (US) 2024-11-28 US claimed
US-20240316208-A1 POLYOXAZOLINE-DRUG CONJUGATES WITH NOVEL PHARMACOKINETIC PROPERTIES SERINA THERAPEUTICS (AL), INC. (US) 2024-09-26 US claimed
US-20020061835-A1 Administering a drug to a human which is pharmaceutically effective to regulate at least one of the blood parameters used to adjust distribution of the drug through the bloodstream RHEOLOGICS, INC. 2002-05-23 US claimed
US-20020032149-A1 Monitoring blood flow parameter of bloodstream, administering substance to organism such that an amount of substance enters bloodstream; distributing portion of amount ofsubstance target within organism RHEOLOGICS, INC. 2002-03-14 US claimed
US-6339716-B1 Method for determining viability of a myocardial segment BIOENERGY INC. 2002-01-15 US claimed
US-20010044584-A1 In vivo delivery methods and compositions RHEOLOGICS, INC. 2001-11-22 US claimed
EP-1098641-A1 CHEMICALLY INDUCED INTRACELLULAR HYPERTHERMIA Texas Pharmaceuticals, Inc. (US) 2001-05-16 EP claimed
WO-2001021218-A2 METHOD FOR DETERMINING VIABILITY OF A MYOCARDIAL SEGMENT BIOENERGY INC. (US) 2001-03-29 WO claimed
EP-1067970-A2 DIAGNOSTIC IMAGING OF VASCULAR ABNORMALITIES USING VASOMODIFICATION NYCOMED IMAGING AS (NO) 2001-01-17 EP claimed
WO-2000006143-A1 CHEMICALLY INDUCED INTRACELLULAR HYPERTHERMIA TEXAS PHARMACEUTICALS, INC. (US) 2000-02-10 WO claimed
WO-1999049899-A2 DIAGNOSTIC IMAGING OF VASCULAR ABNORMALITIES USING VASOMODIFICATION NYCOMED IMAGING AS (NO) 1999-10-07 WO claimed
WO-1992020324-A1 POLYURETHANE HYDROGEL COMPOSITIONS FOR IONTOPHORETIC DRUG DELIVERY GENSIA PHARMACEUTICALS, INC. (US) 1992-11-26 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12383625-B2 Polyoxazoline-drug conjugates with novel pharmacokinetic properties CYP3A5, SPOP, CYP2C19 ADRB2 1728/4885ADRB1 2274/4885ADRB3 1191/4885
US-12485181-B2 Polyoxazoline-drug conjugates with novel pharmacokinetic properties CYP3A5, CYP2C19, CYP3A7 ADRB2 1814/4885ADRB1 2498/4885ADRB3 1120/4885
US-12383626-B2 Polyoxazoline-drug conjugates with novel pharmacokinetic properties CYP3A5, SPOP, CYP2C19 ADRB2 1728/4885ADRB1 2274/4885ADRB3 1191/4885
US-20240316208-A1 POLYOXAZOLINE-DRUG CONJUGATES WITH NOVEL PHARMACOKINETIC PROPERTIES CYP3A5, SPOP, CYP2C19 ADRB2 1728/4885ADRB1 2274/4885ADRB3 1191/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.