SCHEMBL7870515

SCHEMBL7870515

COCCNC(=O)Oc1ccc(C(=O)NS(=O)(=O)c2ccc(CCNC(C)=O)cc2)cn1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.44
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
EGFR P00533 2/20 0.43
ACACB O00763 2/20 0.42
P4HTM Q9NXG6 2/20 0.42
ALDH1A1 P00352 4/20 0.41
EPHX2 P34913 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7862837 0.93 POLB (0.43) POLBMEN1KMT2AEGFRACACB
SCHEMBL7862663 0.91 POLB (0.45) POLBMEN1KMT2AEGFRACACB
SCHEMBL7871648 0.90 RAB9A (0.39) POLBMEN1KMT2AACACBP4HTM
SCHEMBL7870523 0.90 MEN1 (0.47) MEN1KMT2AP4HTMALDH1A1SMN1; SMN2
SCHEMBL7862691 0.90 MEN1 (0.41) POLBMEN1KMT2AEGFRP4HTM
SCHEMBL7862882 0.89 EGFR (0.52) MEN1KMT2AEGFRSMN1; SMN2CA12
SCHEMBL7869432 0.89 EGFR (0.52) MEN1KMT2AEGFRSMN1; SMN2CA12
SCHEMBL7874555 0.89 MAPT (0.51) MEN1KMT2AALDH1A1EPHX2SMN1; SMN2
SCHEMBL7869429 0.89 ALDH1A1 (0.47) POLBMEN1KMT2AEGFRP4HTM
SCHEMBL7871575 0.89 KMT2A (0.56) POLBMEN1KMT2AP4HTMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0562512-B1 Sulfonamidocarbonylpyridine-2-carboxamides and their use as medicines HOECHST AG (DE) 2001-02-21 EP disclosed
EP-0562512-A1 Sulfonamido- and sulfonamidocarbonyl-pyridine-2-carboxamides and their pyridine-N-oxides, process for their preparation and their use as medicines HOECHST AKTIENGESELLSCHAFT (DE) 1993-09-29 EP disclosed