SCHEMBL7874964

SCHEMBL7874964

COC(=O)c1sc(-c2ccccc2)c(-c2ccc(SC)cc2)c1CBr

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 4/20 0.49
TDP1 Q9NUW8 2/20 0.49
NPC1 O15118 2/20 0.49
UBE2N P61088 1/20 0.43
PLA2G1B P04054 1/20 0.39
ATG4B Q9Y4P1 1/20 0.39
TRPM8 Q7Z2W7 1/20 0.38
GRM6 O15303 2/20 0.38
GRIA4 P48058 1/20 0.38
ALDH1A1 P00352 4/20 0.38
KDM4E B2RXH2 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
HPGD P15428 2/20 0.38
HSD17B10 Q99714 1/20 0.38
GRM5 P41594 1/20 0.38
MAPT P10636 3/20 0.36
LMNA P02545 2/20 0.36
TP53 P04637 1/20 0.36
MDM2 Q00987 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7869544 0.90 L3MBTL1 (0.43) L3MBTL1TDP1NPC1UBE2NGRM6
SCHEMBL7876442 0.86 L3MBTL1 (0.43) L3MBTL1TDP1NPC1UBE2NGRIA4
SCHEMBL7869535 0.86 L3MBTL1 (0.47) L3MBTL1TDP1NPC1UBE2NPLA2G1B
SCHEMBL8800287 0.74 GRIA4 (0.49) L3MBTL1TDP1NPC1GRIA4ALDH1A1
SCHEMBL7874913 0.73 PTGS2 (0.49) KDM4EHPGDHSD17B10
SCHEMBL7874918 0.71 NPC1 (0.39) L3MBTL1TDP1NPC1GRM6GRIA4
SCHEMBL8650648 0.69 L3MBTL1 (0.52) L3MBTL1TDP1NPC1UBE2NALDH1A1
SCHEMBL2063437 0.69 ALDH1A1 (0.48) L3MBTL1TDP1PLA2G1BATG4BTRPM8
SCHEMBL7874965 0.68 PTGS1 (0.45) L3MBTL1TDP1NPC1UBE2NGRIA4
SCHEMBL27592419 0.68 ALDH1A1 (0.54) L3MBTL1TDP1PLA2G1BATG4BTRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329421-B1 PHENYL-SUBSTITUTED BENZOFURAN AND BENZOTHIOPHENE DERIVATIVES; NONSTEROIDAL ANTIINFLAMMATORY AGENTS MERCK FROSST CANADA & CO. (CA) 2001-12-11 US disclosed
EP-0778834-B1 DIARYL BICYCLIC HETEROCYCLES AS INHIBITORS OF CYCLOOXYGENASE-2 MERCK FROSST CANADA INC (CA) 2000-01-26 EP disclosed
US-5521213-A NONSTEROID ANTIINFLAMMATORY AGENTS MERCK FROSST CANADA, INC. (CA) 1996-05-28 US disclosed