SCHEMBL787596

SCHEMBL787596

CC1Cc2ccccc2N(C)C1C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.43
HTR2A P28223 5/20 0.41
HTR2C P28335 5/20 0.41
HTR2B P41595 4/20 0.41
ADRA2A P08913 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
ADRA1A P35348 1/20 0.41
HRH1 P35367 1/20 0.41
KCNH2 Q12809 1/20 0.41
OPRM1 P35372 2/20 0.39
PRKCG P05129 1/20 0.38
PRKCA P17252 1/20 0.38
PRKCD Q05655 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21172504 1.00 NOTUM (0.43) NOTUMHTR2AHTR2CHTR2BADRA2A
SCHEMBL21172724 1.00 NOTUM (0.43) NOTUMHTR2AHTR2CHTR2BADRA2A
SCHEMBL12340979 0.89 NOTUM (0.41) NOTUMHTR2AHTR2CHTR2BADRA2A
SCHEMBL21172695 0.81 NOTUM (0.41) NOTUMHTR2AHTR2CHTR2BADRA2A
SCHEMBL7733992 0.79 NOTUM (0.55) NOTUMHTR2AHTR2CHTR2BADRA2A
SCHEMBL6890897 0.79 NOTUM (0.55) NOTUMHTR2AHTR2CHTR2BADRA2A
SCHEMBL31672940 0.79 NOTUM (0.55) NOTUMHTR2AHTR2CHTR2BADRA2A
SCHEMBL811795 0.79 NOTUM (0.55) NOTUMHTR2AHTR2CHTR2BADRA2A
SCHEMBL28217680 0.78 HTR2A (0.44) NOTUMHTR2AHTR2CHTR2BADRA2A
SCHEMBL28217735 0.78 NOTUM (0.42) NOTUMHTR2AHTR2CHTR2BADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0495250-B1 Cationic 1,3,4 thiadiazole dyes BAYER AG (DE) 1996-01-31 EP claimed
EP-0495250-A1 Cationic 1,3,4 thiadiazole dyes BAYER AG (DE) 1992-07-22 EP claimed
US-9748044-B2 Photosensitizer and photoelectric conversion device CHEMICREA INC. (JP) 2017-08-29 US disclosed
US-9703128-B2 Method for making an integrated circuit having optical data communication BrPhotonics Produtos Optoeletronicos LTDA (BR) 2017-07-11 US disclosed
EP-3152306-A1 METHODS AND COMPOUNDS FOR PHOTOTHERAPY WITH CHALCOGENORHODAMINE PHOTOSENSITIZERS Wake Forest University Health Sciences, Inc. (US) 2017-04-12 EP disclosed
US-20170096636-A1 METHODS AND COMPOUNDS FOR PHOTOTHERAPY WITH CHALCOGENORHODAMINE PHOTOSENSITIZERS UNIV WAKE FOREST HEALTH SCIENCES (US) 2017-04-06 US disclosed
US-20170092436-A1 PHOTOSENSITIZER AND PHOTOELECTRIC CONVERSION DEVICE CHEMICREA INC. (JP) 2017-03-30 US disclosed
US-20160349547-A1 METHOD FOR MAKING AN INTEGRATED CIRCUIT HAVING OPTICAL DATA COMMUNICATION LIGHTWAVE LOGIC, INC. 2016-12-01 US disclosed
WO-2015187940-A1 METHODS AND COMPOUNDS FOR PHOTOTHERAPY WITH CHALCOGENORHODAMINE PHOTOSENSITIZERS WAKE FOREST UNIVERSITY HEALTH SCIENCES (US) 2015-12-10 WO disclosed
US-8934741-B2 Integrated circuit with optical data communication Brphotonics Produtos Optoelectronicos LTDA (BR) 2015-01-13 US disclosed
US-20140302250-A1 ELECTRO-OPTIC POLYMER AND ELECTRO-OPTIC DEVICES MADE THEREFROM GIGOPTIX, INC. (US) 2014-10-09 US disclosed
WO-2012037377-A2 INTEGRATED CIRCUIT WITH OPTICAL DATA COMMUNICATION GIGOPTIX, INC. (US) 2012-03-22 WO disclosed
US-20110118232-A1 PYRIMIDINE COMPOUNDS AND USE THEREOF ABBOTT GMBH & CO. KG (DE) 2011-05-19 US disclosed
US-7786105-B2 Pyrimidine compounds and use thereof ABBOTT GMBH & CO. KG (DE) 2010-08-31 US disclosed
US-20090111807-A1 Novel 1,2,3,4-Tetrahydroquinoxaline Derivative Having Glucocorticoid Receptor Binding Activity SANTEN PHARMACEUTICAL CO., LTD. (JP) 2009-04-30 US disclosed
US-20080161322-A1 e.g. 1-[2-tert-Butyl-6-(trifluoromethyl)pyrimidin-4-yl]-4-[3-(2-oxo-3,4-dihydroquinolin-1(2H)-yl)propyl]piperazin-4-ium chloride3,4-Dihydroquinolin-2(1H)-one; dopamine D3 receptor antagonists or agonists; antidepressant, schizophrenia, Parkinson's disease ABBVIE DEUTSCHLAND GMBH & CO KG (DE) 2008-07-03 US disclosed
EP-0495250-B1 Cationic 1,3,4 thiadiazole dyes BAYER AG (DE) 1996-01-31 EP disclosed
US-5208325-A CATIONIC 1,3,4-THIADIAZOLE DYESTUFFS BAYER AKTIENGESELLSCHAFT (DE) 1993-05-04 US disclosed
EP-0495250-A1 Cationic 1,3,4 thiadiazole dyes BAYER AG (DE) 1992-07-22 EP disclosed
US-3991042-A Basic azo dyestuffs containing a benzthiazole and a tetrahydroquinoline nucleus BAYER AKTIENGESELLSCHAFT (DT) 1976-11-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080161322-A1 e.g. 1-[2-tert-Butyl-6-(trifluoromethyl)pyrimidin-4-yl]-4-[3-(2-oxo-3,4-dihydroquinolin-1(2H)-yl)propyl]piperazin-4-ium chloride3,4-Dihydroquinolin-2(1H)-one; dopamine D3 receptor antagonists or agonists; antidepressant, schizophrenia, Parkinson's disease SLC6A3, GRM3, GPR3 NOTUM 4561/4885HTR2A 109/4885HTR2C 49/4885
US-20170096636-A1 METHODS AND COMPOUNDS FOR PHOTOTHERAPY WITH CHALCOGENORHODAMINE PHOTOSENSITIZERS CD4, CD74, NFATC1 NOTUM 2043/4885HTR2A 3808/4885HTR2C 4021/4885
US-20110118232-A1 PYRIMIDINE COMPOUNDS AND USE THEREOF CRHR1, CRHR2, MC2R NOTUM 4351/4885HTR2A 339/4885HTR2C 177/4885
US-20090111807-A1 Novel 1,2,3,4-Tetrahydroquinoxaline Derivative Having Glucocorticoid Receptor Binding Activity NR3C1, NR3C2, MC2R NOTUM 1649/4885HTR2A 568/4885HTR2C 534/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.