Doxribtimine

Doxribtimine

SCHEMBL787714

Cc1cn([C@H]2C[C@H](O)[C@@H](CO)O2)c(=O)[nH]c1=O.Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)n1

nearest known ligand 0.62

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

P

The experimentally established mechanism targets of Doxribtimine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.62
THRB P10828 1/20 0.62
MTOR P42345 1/20 0.62
MDM2 Q00987 1/20 0.62
NCOA1 Q15788 1/20 0.62
NCOA3 Q9Y6Q9 1/20 0.62
P2RY2 P41231 3/20 0.54
P2RY4 P51582 3/20 0.54
P2RY6 Q15077 2/20 0.54
SMN1; SMN2 Q16637 1/20 0.50
TK1 P04183 1/20 0.50
DTYMK P23919 2/20 0.49
TK2 O00142 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Doxribtimine SCHEMBL6518312 1.00 LMNA (0.62) LMNATHRBMTORMDM2NCOA1
Doxribtimine SCHEMBL29124320 0.96 P2RY2 (0.60) LMNATHRBMTORMDM2NCOA1
Doxribtimine SCHEMBL3951759 0.92 TK1 (0.56) LMNASMN1; SMN2TK1TK2
Cytidine SCHEMBL4468985 0.90 LMNA (0.65) LMNATHRBMTORMDM2NCOA1
Adenosine SCHEMBL23835231 0.89 DTYMK (0.66) SMN1; SMN2DTYMK
Cytidine SCHEMBL574775 0.88 LMNA (0.62) LMNATHRBMTORMDM2NCOA1
Guanosine SCHEMBL10528215 0.87 F2 (0.64) LMNATHRBMTORMDM2NCOA1
Cytidine SCHEMBL574822 0.87 LMNA (0.67) LMNATHRBMTORMDM2NCOA1
Doxecitine SCHEMBL9803658 0.87 LMNA (0.50) LMNASMN1; SMN2TK1TK2
Doxribtimine SCHEMBL325199 0.87 TK1 (0.62) LMNASMN1; SMN2TK1TK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20190003966-A1 Ultraviolet and High-Performance Liquid Chromatography Methods for the Evaluation of Sunscreen Efficacy SENA RESEARCH, INCORPORATED (US) 2019-01-03 US claimed
US-20130183765-A1 Ultraviolet and High-Performance Liquid Chromatography Methods for the Evaluation of Sunscreen Efficacy Sena Research Incorporated (US) 2013-07-18 US claimed
WO-2012037158-A2 ULTRAVIOLET AND HIGH-PERFORMANCE LIQUID CHROMATOGRAPHY METHODS FOR THE EVALUATION OF SUNSCREEN EFFICACY SENA RESEARCH, INCORPORATED (US) 2012-03-22 WO claimed
WO-2009027507-A2 APTAMERS WHICH BIND TO A TARGET MOLECULE INVOLVED IN HAEMOSTASIS RHEINISCHE FRIEDRICH-WILHELMS UNIVERSITÄT (DE) 2009-03-05 WO claimed
CN-117016549-B Application of nucleoside compound and composition thereof in promoting plant growth 山东蓬勃生物科技有限公司 2024-02-27 CN disclosed
CN-117016549-A Application of nucleoside compound and composition thereof in promoting plant growth 山东蓬勃生物科技有限公司 2023-11-10 CN disclosed
US-20190003966-A1 Ultraviolet and High-Performance Liquid Chromatography Methods for the Evaluation of Sunscreen Efficacy SENA RESEARCH, INCORPORATED (US) 2019-01-03 US disclosed
US-10073033-B2 Ultraviolet and high-performance liquid chromatography methods for the evaluation of sunscreen efficacy SENA RESEARCH, INC. (US) 2018-09-11 US disclosed
US-20130183765-A1 Ultraviolet and High-Performance Liquid Chromatography Methods for the Evaluation of Sunscreen Efficacy Sena Research Incorporated (US) 2013-07-18 US disclosed
WO-2012037158-A2 ULTRAVIOLET AND HIGH-PERFORMANCE LIQUID CHROMATOGRAPHY METHODS FOR THE EVALUATION OF SUNSCREEN EFFICACY SENA RESEARCH, INCORPORATED (US) 2012-03-22 WO disclosed
US-7700761-B2 3-deoxypentopyranosyl nucleic acid, its production and its use NANOGEN RECOGNOMICS GMBH (DE) 2010-04-20 US disclosed
WO-2009027507-A2 APTAMERS WHICH BIND TO A TARGET MOLECULE INVOLVED IN HAEMOSTASIS RHEINISCHE FRIEDRICH-WILHELMS UNIVERSITÄT (DE) 2009-03-05 WO disclosed
US-20060217546-A1 3-Deoxypentopyranosyl nucleic acid, its production and its use SANOFI (FR) 2006-09-28 US disclosed
EP-1102782-A4 STRUCTURAL ANALOGS OF AMINE BASES AND NUCLEOSIDES BIO RAD LABORATORIES (US) 2002-01-30 EP disclosed
US-6310189-B1 NUCLEOSIDE PHOSPHORAMIDITES OR NUCLEOSIDE H-PHOSPHONATES HAVING A PHOTOREMOVEABLE PROTECTING GROUP COVALENTLY ATTACHED TO A C-3' OR C5' OXYGEN ATOM; PHOTOLITHOGRAPHY; MINIATURIZATION; FINENESS AFFYMETRIX, INC. 2001-10-30 US disclosed
EP-1102782-A1 STRUCTURAL ANALOGS OF AMINE BASES AND NUCLEOSIDES Bio-Rad Laboratories (US) 2001-05-30 EP disclosed
WO-2000008041-A9 STRUCTURAL ANALOGS OF AMINE BASES AND NUCLEOSIDES BIO RAD LABORATORIES (US) 2001-02-01 WO disclosed
WO-2000008041-A1 STRUCTURAL ANALOGS OF AMINE BASES AND NUCLEOSIDES BIO-RAD LABORATORIES (US) 2000-02-17 WO disclosed
US-4788181-A 5-substituted-2',3'-dideoxycytidine compounds with anti-HTLV-III activity THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1988-11-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060217546-A1 3-Deoxypentopyranosyl nucleic acid, its production and its use RNGTT, DTYMK, MTAP LMNA 1658/4885THRB 4486/4885MTOR 2361/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.