SCHEMBL7879563

SCHEMBL7879563

C=CC(=O)NC(C)(C)c1ccc(OCc2ccccc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
KDM4E B2RXH2 2/20 0.52
MEN1 O00255 1/20 0.52
MAPT P10636 1/20 0.52
KMT2A Q03164 1/20 0.52
NPC1 O15118 4/20 0.50
RAB9A P51151 4/20 0.50
CASP3 P42574 1/20 0.50
SENP8 Q96LD8 1/20 0.50
SENP7 Q9BQF6 1/20 0.50
SENP6 Q9GZR1 1/20 0.50
GPR55 Q9Y2T6 1/20 0.50
MAOB P27338 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.48
NR4A2 P43354 2/20 0.48
GSK3B P49841 1/20 0.48
BACE1 P56817 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5396951 0.80 ALDH1A1 (0.58) ALDH1A1CYP3A4CYP2C9CYP2C19MEN1
SCHEMBL5899557 0.78 NPC1 (0.52) ALDH1A1CYP2C19KDM4EMEN1MAPT
SCHEMBL26357615 0.76 LMNA (0.53) ALDH1A1CYP2C19KDM4EMEN1MAPT
SCHEMBL6036170 0.75 MAOB (0.59) CYP2C19KDM4EMEN1MAPTKMT2A
SCHEMBL9020737 0.74 ACACB (0.67) NPC1RAB9AMAOB
Formaldehyde SCHEMBL27841088 0.74 NR4A2 (0.65) CYP2C19KDM4EMEN1MAPTKMT2A
SCHEMBL4677286 0.74 NPC1 (0.57) ALDH1A1CYP2C19KDM4EMEN1MAPT
SCHEMBL5899573 0.74 THRB (0.63) ALDH1A1KDM4EMEN1KMT2ANPC1
SCHEMBL9232869 0.74 PKM (0.59) CYP2C19KDM4EMEN1MAPTKMT2A
SCHEMBL9232872 0.74 PKM (0.59) CYP2C19KDM4EMEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6326500-B1 ANTIINFLAMMATORY AGENTS; ANTIALLERGENS ABBOTT LABORATORIES 2001-12-04 US disclosed
US-6215001-B1 ANTIINFLAMMATORY AGENTS, ANTIASTHMATICS, AND ANTIALLERGENS; SIDE EFFECT REDUCTION KNOLL AKTIENGESELLSCHAFT (DE) 2001-04-10 US disclosed
US-6031109-A Phenoxy-, phenylthio-, benzoyl-alkyleneaminoalkylene-imidazole derivatives as therapeutic agents KNOLL AKTIENGESELLSCHAFT (DE) 2000-02-29 US disclosed
US-5780642-A NON-STEROIDAL ANTIINFLAMMATORY AGENT WHICH BLOCKS RELEASE OF ARACHIDONIC ACID FROM PHOSPHOLIPIDS; SIDE EFFECT REDUCTION KNOLL AKTIENGESELLSCHAFT (DE) 1998-07-14 US disclosed
EP-0705251-A1 IMIDAZOLE DERIVATIVES AS THERAPEUTIC AGENTS Knoll AG (DE) 1996-04-10 EP disclosed
WO-1995000493-A1 IMIDAZOLE DERIVATIVES AS THERAPEUTIC AGENTS KNOLL AG (DE) 1995-01-05 WO disclosed