SCHEMBL7879696

SCHEMBL7879696

COc1ccc(-c2nc3c(o2)CCC(c2ncccc2C2CN2)C3)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.35
RAB9A P51151 4/20 0.35
MAPT P10636 3/20 0.35
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
LMNA P02545 1/20 0.35
ACHE P22303 1/20 0.34
HSP90AA1 P07900 1/20 0.34
PKM P14618 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
GPR119 Q8TDV5 6/20 0.34
TP53 P04637 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
HPGD P15428 1/20 0.34
CYP2C19 P33261 1/20 0.34
AURKA O14965 1/20 0.33
CCNB2 O95067 1/20 0.33
CDK1 P06493 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7880996 0.90 RAB9A (0.43) NPC1RAB9AMAPTALDH1A1KDM4E
SCHEMBL7883808 0.88 GPR119 (0.44) NPC1RAB9AMAPTGPR119CYP1A2
SCHEMBL7877288 0.87 GPR119 (0.36) ALDH1A1ACHEGPR119PRCP
SCHEMBL7882208 0.84 S1PR1 (0.35) NPC1ALDH1A1KDM4EACHEGPR119
SCHEMBL7872792 0.84 S1PR1 (0.35) NPC1ALDH1A1KDM4EACHEGPR119
SCHEMBL7881575 0.83 MAPT (0.36) NPC1RAB9AMAPTALDH1A1KDM4E
SCHEMBL505267 0.83 GRM5 (0.44) NPC1RAB9AMAPTALDH1A1KDM4E
SCHEMBL10250592 0.81 NPC1 (0.45) NPC1RAB9AMAPTALDH1A1KDM4E
SCHEMBL7877057 0.77 GPR119 (0.43) NPC1RAB9AMAPTGPR119CYP1A2
SCHEMBL506208 0.76 NPC1 (0.39) NPC1RAB9AMAPTALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010114971-A1 COMPOUNDS FOR TREATING DISORDERS MEDIATED BY METABOTROPIC GLUTAMATE RECEPTOR 5, AND METHODS OF USE THEREOF SEPRACOR INC. (US) 2010-10-07 WO disclosed