SCHEMBL7885609

SCHEMBL7885609

NC(=O)c1ccc(NC=O)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
L3MBTL1 Q9Y468 2/20 0.47
PARP10 Q53GL7 3/20 0.45
KMT2A Q03164 2/20 0.45
PARP4 Q9UKK3 2/20 0.45
PARP15 Q460N3 1/20 0.45
PARP14 Q460N5 1/20 0.45
PARP16 Q8N5Y8 1/20 0.45
PARP11 Q9NR21 1/20 0.45
KDM4E B2RXH2 1/20 0.45
MAPT P10636 2/20 0.44
PARP1 P09874 2/20 0.44
HSD17B10 Q99714 2/20 0.44
TSHR P16473 2/20 0.44
POLB P06746 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C19 P33261 1/20 0.44
RECQL P46063 1/20 0.44
BLM P54132 1/20 0.44
PMP22 Q01453 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12592838 0.86 ALDH1A1 (0.43) ALDH1A1L3MBTL1PARP10KMT2APARP4
SCHEMBL15453215 0.82 ALDH1A1 (0.52) ALDH1A1L3MBTL1KMT2AMAPTSMN1; SMN2
SCHEMBL4532711 0.82 ALDH1A1 (0.43) ALDH1A1L3MBTL1KMT2AKDM4EMAPT
SCHEMBL7440442 0.81 PRSS1 (0.57) ALDH1A1HSD17B10CYP2C19F2PRSS1
SCHEMBL1086165 0.80 ALDH1A1 (0.56) ALDH1A1KMT2AKDM4ETSHRSMN1; SMN2
SCHEMBL4795623 0.79 ALDH1A1 (0.44) ALDH1A1L3MBTL1PARP10KMT2APARP4
SCHEMBL1086084 0.78 ALDH1A1 (0.54) ALDH1A1KMT2AKDM4ETSHRSMN1; SMN2
SCHEMBL3691518 0.78 ALDH1A1 (0.38) ALDH1A1L3MBTL1PARP10KMT2APARP15
SCHEMBL14705725 0.78 PEPD (0.59) ALDH1A1KMT2AMAPTHSD17B10CA2
SCHEMBL1555352 0.78 MAPT (0.54) ALDH1A1L3MBTL1KMT2AKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0912574-A1 BETA-LACTAMS F. HOFFMANN-LA ROCHE AG (CH) 1999-05-06 EP claimed
WO-1997045429-A1 BETA-LACTAMS F. HOFFMANN-LA ROCHE AG (CH) 1997-12-04 WO claimed
US-5494666-A BETA-LACTAMASE INHIBITORS, ANTIBACTERIALS HOFFMANN-LA ROCHE INC. (US) 1996-02-27 US claimed
US-5464617-A 1H-2,6a-diazacyclobut(cd)indene-6-carboxylic acid derivatives, antibiotics HOFFMANN-LA ROCHE INC. (US) 1995-11-07 US claimed
US-20230348441-A1 BICYCLIC COMPOUND THAT ACTS AS CRBN PROTEIN REGULATOR MEDSHINE DISCOVERY INC. (CN) 2023-11-02 US disclosed
CN-112125828-B Synthetic method of foramsulfuron intermediate 江苏省农用激素工程技术研究中心有限公司 2022-05-06 CN disclosed
WO-2021047674-A1 BICYCLIC COMPOUND THAT ACTS AS CRBN PROTEIN REGULATOR 南京明德新药研发有限公司 2021-03-18 WO disclosed
CN-105670340-B Preparation method of C.I. pigment yellow 180 上虞市新利化工有限公司 2017-05-03 CN disclosed
CN-100500654-C Tetrahydrocarbazole derivatives as ligands for G-protein coupled receptors (GPCRs) ZENTARIS AG (DE) 2009-06-17 CN disclosed
US-20070232654-A1 Novel Compounds and Compositions as Cathepsin Inhibitors AXYS PHARMACEUTICALS, INC. (US) 2007-10-04 US disclosed
CN-1599720-A Tetrahydrocarbazole derivatives as ligands for G-protein coupled receptors (GPCRs) ZENTARIS AG (DE) 2005-03-23 CN disclosed
US-6218379-B1 Tricyclic carbacephems HOFFMANN-LA ROCHE INC. 2001-04-17 US disclosed
US-5633282-A ENZYME INHIBITORS BRITISH TECHNOLOGY GROUP LIMITED (GB) 1997-05-27 US disclosed
EP-0531370-B1 INHIBITION OF VIRAL INFECTION BRITISH TECH GROUP (GB) 1996-09-18 EP disclosed
US-5494666-A BETA-LACTAMASE INHIBITORS, ANTIBACTERIALS HOFFMANN-LA ROCHE INC. (US) 1996-02-27 US disclosed
US-5464617-A 1H-2,6a-diazacyclobut(cd)indene-6-carboxylic acid derivatives, antibiotics HOFFMANN-LA ROCHE INC. (US) 1995-11-07 US disclosed
EP-0671401-A1 Beta lactames F. HOFFMANN-LA ROCHE AG (CH) 1995-09-13 EP disclosed
EP-0531370-A1 INHIBITION OF VIRAL INFECTION. COLLINS MARY KATHARINE LEVINGE (GB) 1993-03-17 EP disclosed
WO-1991018591-A1 INHIBITION OF VIRAL INFECTION COLLINS MARY KATHARINE LEVINGE (GB) 1991-12-12 WO disclosed
US-5026831-A Water-insoluble disazo colorants having hetero-bicyclic methylene-active compounds as coupling component HOECHST AKTIENGESELLSCHAFT (DE) 1991-06-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230348441-A1 BICYCLIC COMPOUND THAT ACTS AS CRBN PROTEIN REGULATOR CRBN, CRKL, NCOR1 ALDH1A1 4261/4885L3MBTL1 4032/4885PARP10 3256/4885
US-20070232654-A1 Novel Compounds and Compositions as Cathepsin Inhibitors CTSS, CTSB, CTSE ALDH1A1 4046/4885L3MBTL1 4113/4885PARP10 2228/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.