SCHEMBL789053

SCHEMBL789053

CS(=O)(=O)c1cc(F)c(N[C@@H]2CNCCC2N2CCCC2=O)cc1F

nearest known ligand 0.32

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 7/20 0.32
IRAK4 Q9NWZ3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL789678 0.96 SCN9A (0.33) SCN9A
SCHEMBL2597088 0.93 F10 (0.31) IRAK4
SCHEMBL789216 0.86 SLC6A9 (0.34) IRAK4
SCHEMBL789299 0.83 DPP4 (0.30)
SCHEMBL2597109 0.83 SLC6A9 (0.37)
SCHEMBL790391 0.81 BRD4 (0.33)
SCHEMBL790469 0.80 SCN9A (0.34) SCN9A
SCHEMBL788886 0.80 SCN9A (0.34) SCN9A
SCHEMBL789443 0.75 AKR1C3 (0.34)
SCHEMBL797320 0.72 BTK (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616074-A1 PIPERIDINYL-SUBSTITUTED LACTAMS AS GPR119 MODULATORS Array Biopharma, Inc. (US) 2013-07-24 EP disclosed
EP-2571864-A1 PIPERIDINYL-SUBSTITUTED LACTAMS AS GPR119 MODULATORS Array Biopharma, Inc. (US) 2013-03-27 EP disclosed
WO-2012037393-A1 PIPERIDINYL-SUBSTITUTED LACTAMS AS GPR119 MODULATORS ARRAY BIOPHARMA INC. (US) 2012-03-22 WO disclosed
WO-2011146335-A1 PIPERIDINYL-SUBSTITUTED LACTAMS AS GPR119 MODULATORS ARRAY BIOPHARMA INC. (US) 2011-11-24 WO disclosed