SCHEMBL789220

SCHEMBL789220

Cc1sc(Nc2ccc3c(c2)OCCO3)nc1C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.53
ALDH1A1 P00352 5/20 0.53
SMN1; SMN2 Q16637 4/20 0.53
NPC1 O15118 4/20 0.53
RAB9A P51151 4/20 0.53
GLA P06280 1/20 0.53
HPGD P15428 1/20 0.53
TRPC3 Q13507 2/20 0.52
TRPC6 Q9Y210 2/20 0.52
DHODH Q02127 1/20 0.48
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
LMNA P02545 2/20 0.47
GAA P10253 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2C19 P33261 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
HTT P42858 1/20 0.45
HSD17B10 Q99714 2/20 0.45
TSHR P16473 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14184605 0.83 RAB9A (0.53) MAPTALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL10087862 0.81 TRPC3 (0.60) MAPTALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL806599 0.77 TRPC3 (0.58) MAPTALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL2873347 0.76 ALDH1A1 (0.50) MAPTALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL16586316 0.76 GAA (0.63) MAPTALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL2877955 0.75 DHODH (0.55) MAPTALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL19667972 0.72 NPC1 (0.40) MAPTALDH1A1NPC1RAB9AHPGD
SCHEMBL22053468 0.72 GAA (0.40) MAPTALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL2878623 0.72 MAPT (0.44) MAPTALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL807014 0.72 TRPC3 (0.73) MAPTALDH1A1SMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037349-A2 COMPOUNDS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed
WO-2012037351-A1 COMPOUNDS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed
WO-2012037351-A1 COMPOUNDS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed