SCHEMBL789385

SCHEMBL789385

N#Cc1c(-c2ccc(C(=O)N3CCOCC3)cc2)c(N)nc2ccc(-c3cnc(N)c(S(=O)(=O)NC4CC4)c3)cc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BMPR1B O00238 3/20 0.45
BMPR1A P36894 3/20 0.45
ACVRL1 P37023 3/20 0.45
ACVR1 Q04771 3/20 0.45
TGFBR1 P36897 2/20 0.45
KCNH2 Q12809 3/20 0.41
JAK2 O60674 1/20 0.40
LIPC P11150 2/20 0.39
LIPG Q9Y5X9 2/20 0.39
ATR Q13535 2/20 0.39
PIK3CD O00329 1/20 0.38
PIK3R1 P27986 1/20 0.38
LRRK2 Q5S007 1/20 0.38
TBK1 Q9UHD2 1/20 0.38
CSF1R P07333 1/20 0.37
PIK3CA P42336 1/20 0.37
SFRP1 Q8N474 1/20 0.37
HPGD P15428 1/20 0.37
MET P08581 1/20 0.37
NTRK1 P04629 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL807212 0.82 PIK3CD (0.46) KCNH2JAK2PIK3CDPIK3R1LRRK2
SCHEMBL807280 0.81 PIK3CD (0.50) KCNH2PIK3CDPIK3R1CSF1RPIK3CA
SCHEMBL806789 0.79 PIK3CD (0.50) BMPR1BBMPR1AACVRL1ACVR1TGFBR1
SCHEMBL789847 0.77 JAK2 (0.46) KCNH2JAK2ATRPIK3CDPIK3CA
SCHEMBL14247596 0.69 BMPR1B (0.44) BMPR1BBMPR1AACVRL1ACVR1TGFBR1
SCHEMBL807223 0.67 IRAK4 (0.46) BMPR1BBMPR1AACVRL1ACVR1TGFBR1
SCHEMBL14247756 0.67 BRD4 (0.44) BMPR1BBMPR1AACVRL1ACVR1TGFBR1
SCHEMBL14317285 0.66 BMPR1B (0.43) BMPR1BBMPR1AACVRL1ACVR1TGFBR1
SCHEMBL9954675 0.66 PI4KA (0.61)
SCHEMBL14247512 0.66 PIK3CB (0.42) KCNH2ATRPIK3CDPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed