SCHEMBL806789

SCHEMBL806789

COc1ncc(-c2ccc3nc(N)c(-c4ccc(C(=O)N5CCOCC5)cc4)c(C#N)c3c2)cc1N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 7/20 0.50
PIK3R1 P27986 1/20 0.50
IRAK4 Q9NWZ3 1/20 0.45
KIT P10721 1/20 0.44
JAK2 O60674 1/20 0.43
LRRK2 Q5S007 2/20 0.43
PIK3CA P42336 5/20 0.43
PIK3CG P48736 5/20 0.43
PIK3CB P42338 4/20 0.43
KCNH2 Q12809 3/20 0.43
MTOR P42345 1/20 0.41
NTRK1 P04629 1/20 0.40
BMPR1B O00238 1/20 0.40
BMPR1A P36894 1/20 0.40
TGFBR1 P36897 1/20 0.40
ACVRL1 P37023 1/20 0.40
ACVR1 Q04771 1/20 0.40
ATR Q13535 1/20 0.40
HPGD P15428 2/20 0.40
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL807223 0.88 IRAK4 (0.46) PIK3CDPIK3R1IRAK4KITJAK2
SCHEMBL807212 0.87 PIK3CD (0.46) PIK3CDPIK3R1KITJAK2LRRK2
SCHEMBL807280 0.86 PIK3CD (0.50) PIK3CDPIK3R1PIK3CAPIK3CGPIK3CB
SCHEMBL789847 0.81 JAK2 (0.46) PIK3CDJAK2PIK3CAKCNH2MTOR
SCHEMBL789385 0.79 BMPR1B (0.45) PIK3CDPIK3R1JAK2LRRK2PIK3CA
SCHEMBL10277093 0.79 KDM4E (0.43) PIK3CDIRAK4PIK3CAPIK3CGPIK3CB
SCHEMBL806763 0.77 KIT (0.49) PIK3CDPIK3R1IRAK4KITLRRK2
SCHEMBL789702 0.72 PIK3CG (0.52) PIK3CDPIK3R1PIK3CAPIK3CGPIK3CB
SCHEMBL789701 0.72 PIK3CG (0.73) PIK3CDPIK3R1PIK3CAPIK3CGPIK3CB
SCHEMBL807275 0.71 PIK3CG (0.63) PIK3CDPIK3R1PIK3CAPIK3CGPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed