SCHEMBL789847

SCHEMBL789847

N#Cc1c(-c2ccc(C(=O)N3CCOCC3)cc2)c(N)nc2ccc(I)cc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.46
HPGD P15428 4/20 0.42
ATR Q13535 1/20 0.42
ADORA2A P29274 1/20 0.41
PDCD1 Q15116 1/20 0.41
CD274 Q9NZQ7 1/20 0.41
KCNH2 Q12809 3/20 0.40
MKNK1 Q9BUB5 3/20 0.40
MKNK2 Q9HBH9 3/20 0.40
CDK1 P06493 1/20 0.40
EIF4E P06730 1/20 0.40
GRM2 Q14416 1/20 0.40
PIK3CD O00329 1/20 0.39
PIK3CA P42336 1/20 0.39
MTOR P42345 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HDAC4 P56524 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL790084 0.85 JAK2 (0.48) JAK2HPGDATRKCNH2MKNK1
SCHEMBL790839 0.85 ADORA2A (0.49) HPGDADORA2ACDK1KDM4EALDH1A1
SCHEMBL806789 0.81 PIK3CD (0.50) JAK2HPGDATRKCNH2PIK3CD
SCHEMBL789385 0.77 BMPR1B (0.45) JAK2HPGDATRKCNH2PIK3CD
SCHEMBL790759 0.76 KDM4E (0.47) HPGDADORA2APIK3CDPIK3CAKDM4E
SCHEMBL807212 0.75 PIK3CD (0.46) JAK2KCNH2PIK3CDPIK3CAMTOR
SCHEMBL807280 0.74 PIK3CD (0.50) KCNH2PIK3CDPIK3CAMTORALDH1A1
SCHEMBL10277681 0.72 LRRK2 (0.47) JAK2ATRKDM4EALDH1A1SMN1; SMN2
SCHEMBL790716 0.69 MAPT (0.43) HPGDADORA2AKDM4EALDH1A1SMN1; SMN2
SCHEMBL109082 0.69 PHGDH (0.69) HPGDKDM4EALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed