SCHEMBL7900184

SCHEMBL7900184

COC(=O)CCNC(=O)c1cccc(N)c1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 1/20 0.53
CTSG P08311 1/20 0.53
CTRB1 P17538 1/20 0.53
CMA1 P23946 1/20 0.53
SMN1; SMN2 Q16637 3/20 0.51
MAPT P10636 2/20 0.51
ALDH1A1 P00352 2/20 0.50
KDM4E B2RXH2 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
MAPK1 P28482 1/20 0.45
NPSR1 Q6W5P4 1/20 0.44
HSD17B10 Q99714 1/20 0.44
MAPK14 Q16539 1/20 0.44
LMNA P02545 1/20 0.44
HTT P42858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4955045 0.92 MAPT (0.54) SMN1; SMN2MAPTALDH1A1KDM4EMEN1
SCHEMBL7145528 0.86 PRSS1 (0.48) PRSS1CTSGCTRB1CMA1SMN1; SMN2
SCHEMBL2299009 0.85 HPGD (0.59) SMN1; SMN2ALDH1A1KDM4EL3MBTL1
SCHEMBL6160025 0.85 MAPK1 (0.60) SMN1; SMN2ALDH1A1KDM4EMEN1KMT2A
SCHEMBL10630944 0.84 ALDH1A1 (0.57) SMN1; SMN2ALDH1A1KDM4EL3MBTL1MEN1
SCHEMBL27371604 0.83 ITGB3 (0.54) PRSS1CTSGCTRB1CMA1SMN1; SMN2
SCHEMBL277398 0.83 KDM4E (0.50) PRSS1CTSGCTRB1CMA1SMN1; SMN2
SCHEMBL12497737 0.82 ALDH1A1 (0.64) SMN1; SMN2MAPTALDH1A1KDM4E
SCHEMBL658648 0.81 L3MBTL1 (0.69) SMN1; SMN2ALDH1A1KDM4EL3MBTL1KMT2A
SCHEMBL2667533 0.81 LMNA (0.56) PRSS1CTSGCTRB1CMA1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0608759-B1 Piperazine derivatives MERCK PATENT GMBH (DE) 2001-08-22 EP disclosed
US-5908843-A Piperazine compounds as fibrinogen inhibitors MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1999-06-01 US disclosed
EP-0608759-A2 Piperazinderivatives MERCK PATENT GmbH (DE) 1994-08-03 EP disclosed