SCHEMBL277398

SCHEMBL277398

NC(=O)CCNC(=O)c1cccc(N)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
SMN1; SMN2 Q16637 2/20 0.49
HSD17B10 Q99714 2/20 0.48
NPSR1 Q6W5P4 1/20 0.48
KDM4C Q9H3R0 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.46
PRMT5 O14744 1/20 0.46
WDR77 Q9BQA1 1/20 0.46
PBRM1 Q86U86 1/20 0.46
PRSS1 P07477 2/20 0.45
CTSG P08311 1/20 0.45
CTRB1 P17538 1/20 0.45
CMA1 P23946 1/20 0.45
PTGS1 P23219 1/20 0.44
HDAC1 Q13547 4/20 0.44
HDAC3 O15379 3/20 0.44
LMNA P02545 1/20 0.43
F2 P00734 1/20 0.43
PLG P00747 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10630944 0.88 ALDH1A1 (0.57) KDM4EALDH1A1SMN1; SMN2HSD17B10NPSR1
SCHEMBL27371604 0.87 ITGB3 (0.54) KDM4EALDH1A1SMN1; SMN2HSD17B10NPSR1
SCHEMBL12516004 0.85 SMN1; SMN2 (0.62) KDM4EALDH1A1SMN1; SMN2HSD17B10NPSR1
SCHEMBL11118792 0.84 HDAC6 (0.54) KDM4EALDH1A1SMN1; SMN2HSD17B10NPSR1
SCHEMBL10123874 0.83 TERT (0.55) KDM4EALDH1A1SMN1; SMN2HSD17B10NPSR1
SCHEMBL3650167 0.83 HPGD (0.54) KDM4EALDH1A1SMN1; SMN2HSD17B10NPSR1
SCHEMBL8298056 0.83 KDM4E (0.53) KDM4EALDH1A1SMN1; SMN2HSD17B10NPSR1
Hydrochloric Acid SCHEMBL10771309 0.83 HDAC6 (0.52) KDM4EALDH1A1SMN1; SMN2HSD17B10NPSR1
SCHEMBL7900184 0.83 PRSS1 (0.53) KDM4EALDH1A1SMN1; SMN2HSD17B10NPSR1
SCHEMBL279941 0.83 RAB9A (0.62) KDM4EALDH1A1SMN1; SMN2HSD17B10HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8134013-B2 Amide compound and thrombopoietin receptor activator NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2012-03-13 US disclosed
US-20090131659-A1 AMIDE COMPOUND AND THROMBOPOIETIN RECEPTOR ACTIVATOR NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2009-05-21 US disclosed
CN-101076519-A Amide compound and thrombopoietin receptor activator NISSAN CHEMICAL IND LTD (JP) 2007-11-21 CN disclosed
EP-1845090-A1 AMIDE COMPOUND AND THROMBOPOIETIN RECEPTOR ACTIVATOR Nissan Chemical Industries, Ltd. (JP) 2007-10-17 EP disclosed
US-6858641-B2 Substituted indolinones BOEHRINGER INGELHEIM PHARMA KG (DE) 2005-02-22 US disclosed
CN-1509270-A Indolinones substituted in the 6-position, process for their preparation and their use as kinase inhibitors ���ָ��Ӣ��ķ�������Ϲ�˾ 2004-06-30 CN disclosed
EP-1379501-A1 INDOLINONES, SUBSTITUTED IN POSITION 6, AND THEIR USE AS KINASE INHIBITORS Boehringer Ingelheim Pharma GmbH & Co.KG (DE) 2004-01-14 EP disclosed
US-20030092756-A1 Substituted indolinones BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2003-05-15 US disclosed
WO-2002081445-A1 INDOLINONES, SUBSTITUTED IN POSITION 6, AND THEIR USE AS KINASE INHIBITORS BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2002-10-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030092756-A1 Substituted indolinones CDK1, CDK2, CDKL1 KDM4E 695/4885ALDH1A1 1526/4885SMN1; SMN2 4355/4885
US-20090131659-A1 AMIDE COMPOUND AND THROMBOPOIETIN RECEPTOR ACTIVATOR TEK, PTAFR, MPL KDM4E 4435/4885ALDH1A1 2047/4885SMN1; SMN2 1437/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.